SCHEMBL807541

SCHEMBL807541

CC(C)(C)OC(=O)N1CCC(Nc2cc(CN3CCOCC3)cc(Nc3nc4cccnc4s3)n2)CC1

nearest known ligand 0.55

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ITK Q08881 2/20 0.55
SSTR5 P35346 1/20 0.46
TBK1 Q9UHD2 14/20 0.45
RORC P51449 1/20 0.43
DHODH Q02127 1/20 0.43
LCK P06239 1/20 0.42
AURKB Q96GD4 1/20 0.42
CCNA2 P20248 1/20 0.41
CDK2 P24941 1/20 0.41
SYK P43405 1/20 0.40
IKBKE Q14164 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL807926 0.96 ITK (0.59) ITKSSTR5TBK1RORCDHODH
SCHEMBL807803 0.87 ITK (0.58) ITKSSTR5TBK1RORCDHODH
SCHEMBL807714 0.85 ITK (0.46) ITKSSTR5TBK1RORCDHODH
SCHEMBL793964 0.84 ITK (0.56) ITKSSTR5RORCDHODHLCK
SCHEMBL2398982 0.84 ITK (0.57) ITKSSTR5RORCDHODHLCK
SCHEMBL2398991 0.84 ITK (0.57) ITKSSTR5RORCDHODHLCK
SCHEMBL807822 0.80 ITK (0.81) ITKSSTR5RORCDHODHLCK
SCHEMBL807716 0.80 ITK (0.60) ITKRORCDHODHLCKAURKB
SCHEMBL807721 0.80 KMT2A (0.49) ITKTBK1LCKAURKB
SCHEMBL808081 0.79 ITK (0.54) ITKSSTR5TBK1RORCDHODH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012035055-A1 NOVEL COMPOUNDS GLAXO GROUP LIMITED (GB) 2012-03-22 WO disclosed