SCHEMBL807714

SCHEMBL807714

CC(C)(C)OC(=O)N1CCC(Nc2cc(CN3CCOCC3)cc(Nc3nc4ccccc4s3)n2)C1

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ITK Q08881 2/20 0.46
SSTR5 P35346 4/20 0.44
BRD4 O60885 1/20 0.42
RAB9A P51151 2/20 0.41
BTK Q06187 2/20 0.41
LCK P06239 1/20 0.41
NPC1 O15118 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
LTA4H P09960 1/20 0.41
KCNH2 Q12809 1/20 0.41
HCK P08631 1/20 0.40
DHODH Q02127 5/20 0.40
RORC P51449 4/20 0.40
TBK1 Q9UHD2 1/20 0.40
KDM1A O60341 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL807721 0.90 KMT2A (0.49) ITKRAB9ALCKNPC1TBK1
SCHEMBL807926 0.89 ITK (0.59) ITKSSTR5BRD4BTKLCK
SCHEMBL807541 0.85 ITK (0.55) ITKSSTR5LCKDHODHRORC
SCHEMBL807803 0.80 ITK (0.58) ITKSSTR5BRD4BTKLCK
SCHEMBL23608014 0.80 BTK (0.42) ITKBRD4BTKHCKTBK1
SCHEMBL21792649 0.80 BTK (0.42) ITKBRD4BTKHCKTBK1
SCHEMBL798203 0.79 ITK (0.42) ITKSSTR5RAB9ALCKNPC1
SCHEMBL21792590 0.79 BTK (0.41) ITKBTKHCKTBK1
SCHEMBL29261762 0.79 BTK (0.41) ITKBTKHCKTBK1
SCHEMBL10285559 0.79 KMT2A (0.51) ITKRAB9ABTKLCKNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012035055-A1 NOVEL COMPOUNDS GLAXO GROUP LIMITED (GB) 2012-03-22 WO disclosed