SCHEMBL8077802

SCHEMBL8077802

CC(=N)NCCCCC(N)c1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 1/20 0.41
MTNR1B P49286 1/20 0.41
KDM1A O60341 3/20 0.39
NAAA Q02083 2/20 0.39
MAOB P27338 2/20 0.39
HTR2A P28223 1/20 0.38
HRH1 P35367 1/20 0.38
SIGMAR1 Q99720 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8077419 0.86 SLC2A1 (0.36)
Hydrochloric Acid SCHEMBL8080750 0.81 ALDH1A1 (0.41) MTNR1AMTNR1BKDM1ANAAAMAOB
SCHEMBL10324528 0.81 NAAA (0.44) MTNR1AMTNR1BKDM1ANAAAMAOB
SCHEMBL8077823 0.81 TSHR (0.37) NAAA
SCHEMBL17373052 0.77 SCN4A (0.50) HTR2AHRH1
SCHEMBL3509613 0.76 MTNR1A (0.45) MTNR1AMTNR1BNAAA
Hydrochloric Acid SCHEMBL28350804 0.75 SCN4A (0.48) HTR2AHRH1
SCHEMBL10324521 0.75 MEN1 (0.54) MAOB
SCHEMBL8421133 0.72 MTNR1A (0.72) MTNR1AMTNR1B
SCHEMBL869237 0.72 SLC2A1 (0.57) HTR2AHRH1SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6143790-A ENZYME INHIBITORS G.D. SEARLE & CO. (US) 2000-11-07 US claimed
WO-1995024382-A1 L-N6-(1-IMINOETHYL)LYSINE DERIVATIVES USEFUL AS NITRIC OXIDE SYNTHASE INHIBITORS G.D. SEARLE & CO. (US) 1995-09-14 WO claimed
US-6143790-A ENZYME INHIBITORS G.D. SEARLE & CO. (US) 2000-11-07 US disclosed
EP-0749418-B1 L-N6 -(1-IMINOETHYL)LYSINE DERIVATIVES USEFUL AS NITRIC OXIDE SYNTHASE INHIBITORS SEARLE & CO (US) 2000-08-30 EP disclosed
WO-1995024382-A1 L-N6-(1-IMINOETHYL)LYSINE DERIVATIVES USEFUL AS NITRIC OXIDE SYNTHASE INHIBITORS G.D. SEARLE & CO. (US) 1995-09-14 WO disclosed