SCHEMBL807802

SCHEMBL807802

COCc1cc(Nc2nc3cccnc3s2)nc(NCCCCN)n1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.47
LCK P06239 4/20 0.45
ITK Q08881 4/20 0.45
AURKB Q96GD4 4/20 0.45
POLB P06746 1/20 0.42
HSP90AA1 P07900 2/20 0.38
HSP90AB1 P08238 2/20 0.38
RAB9A P51151 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
RAD52 P43351 1/20 0.35
MEN1 O00255 1/20 0.34
ALDH1A1 P00352 1/20 0.34
TP53 P04637 1/20 0.34
HTT P42858 1/20 0.34
KMT2A Q03164 1/20 0.34
SSTR5 P35346 1/20 0.34
SYK P43405 4/20 0.33
CHEK1 O14757 1/20 0.33
CDK7 P50613 1/20 0.33
TXK P42681 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10286441 0.93 ITK (0.47) NPC1LCKITKAURKBPOLB
SCHEMBL12470060 0.85 LCK (0.47) NPC1LCKITKAURKBPOLB
SCHEMBL808038 0.85 LCK (0.46) NPC1LCKITKAURKBPOLB
SCHEMBL793708 0.78 LCK (0.40) NPC1LCKITKAURKBPOLB
SCHEMBL799038 0.76 POLB (0.44) NPC1LCKITKAURKBPOLB
SCHEMBL807804 0.71 LCK (0.46) NPC1LCKITKAURKBPOLB
SCHEMBL12291456 0.69 NPC1 (0.44) NPC1LCKITKAURKBPOLB
SCHEMBL136795 0.66 LCK (0.66) NPC1LCKITKAURKBRAB9A
SCHEMBL19792489 0.66 NPC1 (0.89) NPC1POLBRAB9ASMN1; SMN2ALDH1A1
SCHEMBL139646 0.66 ITK (0.69) LCKITKAURKBSSTR5TXK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012035055-A1 NOVEL COMPOUNDS GLAXO GROUP LIMITED (GB) 2012-03-22 WO disclosed