SCHEMBL793708

SCHEMBL793708

COCc1cc(Nc2nc3cccnc3s2)nc(NCC/C(=C\CN(C)C)C(N)=O)n1

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
LCK P06239 5/20 0.40
ITK Q08881 4/20 0.40
AURKB Q96GD4 3/20 0.40
NPC1 O15118 2/20 0.35
POLB P06746 1/20 0.35
RAB9A P51151 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
BUB1 O43683 1/20 0.32
SSTR5 P35346 1/20 0.30
FYN P06241 1/20 0.30
SRC P12931 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10286441 0.80 ITK (0.47) LCKITKAURKBNPC1POLB
SCHEMBL808038 0.80 LCK (0.46) LCKITKAURKBNPC1POLB
SCHEMBL12470060 0.80 LCK (0.47) LCKITKAURKBNPC1POLB
SCHEMBL807802 0.78 NPC1 (0.47) LCKITKAURKBNPC1POLB
SCHEMBL799038 0.70 POLB (0.44) LCKITKAURKBNPC1POLB
SCHEMBL10285615 0.69 LCK (0.40) LCKITKAURKBNPC1POLB
SCHEMBL807917 0.65 LCK (0.39) LCKITKAURKBNPC1POLB
SCHEMBL145043 0.63 ITK (0.68) LCKITKAURKBSSTR5SRC
SCHEMBL145042 0.63 ITK (0.68) LCKITKAURKBSSTR5SRC
SCHEMBL807804 0.63 LCK (0.46) LCKITKAURKBNPC1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012035055-A1 NOVEL COMPOUNDS GLAXO GROUP LIMITED (GB) 2012-03-22 WO disclosed