SCHEMBL807804

SCHEMBL807804

CNCCNc1nc(CN2CCOCC2)cc(Nc2nc3cccnc3s2)n1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LCK P06239 6/20 0.46
ITK Q08881 3/20 0.46
AURKB Q96GD4 2/20 0.46
POLB P06746 1/20 0.40
NPC1 O15118 2/20 0.39
HCK P08631 2/20 0.38
BTK Q06187 2/20 0.38
RORC P51449 1/20 0.37
DHODH Q02127 1/20 0.37
IGF1R P08069 1/20 0.37
SSTR5 P35346 1/20 0.37
PIK3CD O00329 1/20 0.36
PIK3CA P42336 1/20 0.36
PIK3CB P42338 1/20 0.36
PIK3CG P48736 1/20 0.36
CXCR4 P61073 1/20 0.36
RAB9A P51151 2/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
KDR P35968 1/20 0.35
MEN1 O00255 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10285615 0.83 LCK (0.40) LCKITKAURKBPOLBNPC1
SCHEMBL807917 0.82 LCK (0.39) LCKITKAURKBPOLBNPC1
SCHEMBL139140 0.81 LCK (0.70) LCKITKAURKBHCKBTK
SCHEMBL139139 0.81 LCK (0.70) LCKITKAURKBHCKBTK
SCHEMBL10286653 0.79 HCK (0.44) LCKITKAURKBHCKBTK
SCHEMBL111924 0.77 AURKB (0.55) LCKITKAURKBHCKBTK
SCHEMBL24019194 0.75 KDR (0.44) LCKITKAURKBPOLBNPC1
SCHEMBL798710 0.75 LCK (0.45) LCKITKAURKBPOLBNPC1
SCHEMBL807713 0.73 ITK (0.41) LCKITKAURKBPOLBNPC1
SCHEMBL138604 0.73 ITK (0.71) LCKITKAURKBBTKRORC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012035055-A1 NOVEL COMPOUNDS GLAXO GROUP LIMITED (GB) 2012-03-22 WO disclosed