SCHEMBL807917

SCHEMBL807917

CN(CCNc1nc(CN2CCOCC2)cc(Nc2nc3cccnc3s2)n1)C(=O)OC(C)(C)C

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LCK P06239 5/20 0.39
ITK Q08881 2/20 0.39
AURKB Q96GD4 1/20 0.39
RORC P51449 1/20 0.38
DHODH Q02127 1/20 0.38
HCK P08631 2/20 0.37
BTK Q06187 2/20 0.37
AAK1 Q2M2I8 1/20 0.34
PIK3CD O00329 1/20 0.34
PIK3CA P42336 1/20 0.34
PIK3CB P42338 1/20 0.34
PIK3CG P48736 1/20 0.34
JAK2 O60674 1/20 0.33
JAK3 P52333 1/20 0.33
KCNH2 Q12809 1/20 0.33
SSTR5 P35346 1/20 0.33
NPC1 O15118 1/20 0.33
POLB P06746 1/20 0.33
CXCR4 P61073 1/20 0.32
RAB9A P51151 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL807804 0.82 LCK (0.46) LCKITKAURKBRORCDHODH
SCHEMBL10285615 0.80 LCK (0.40) LCKITKAURKBRORCDHODH
SCHEMBL807713 0.77 ITK (0.41) LCKITKAURKBRORCDHODH
SCHEMBL808049 0.76 LCK (0.43) LCKRORCDHODHHCKBTK
SCHEMBL10286653 0.76 HCK (0.44) LCKITKAURKBRORCDHODH
SCHEMBL139140 0.74 LCK (0.70) LCKITKAURKBRORCDHODH
SCHEMBL139139 0.74 LCK (0.70) LCKITKAURKBRORCDHODH
SCHEMBL807541 0.72 ITK (0.55) LCKITKAURKBRORCDHODH
SCHEMBL807926 0.71 ITK (0.59) LCKITKAURKBRORCDHODH
SCHEMBL111924 0.69 AURKB (0.55) LCKITKAURKBRORCDHODH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012035055-A1 NOVEL COMPOUNDS GLAXO GROUP LIMITED (GB) 2012-03-22 WO disclosed