SCHEMBL798710

SCHEMBL798710

Clc1cc(CN2CCOCC2)cc(Nc2nc3cccnc3s2)n1

nearest known ligand 0.45

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
LCK P06239 6/20 0.45
RAB9A P51151 2/20 0.44
KDR P35968 1/20 0.44
NPC1 O15118 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
SSTR5 P35346 1/20 0.44
ITK Q08881 2/20 0.43
AURKB Q96GD4 1/20 0.43
POLB P06746 1/20 0.40
EGFR P00533 2/20 0.39
RORC P51449 1/20 0.39
DHODH Q02127 1/20 0.39
LTA4H P09960 4/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24019194 0.88 KDR (0.44) LCKRAB9AKDRNPC1SMN1; SMN2
SCHEMBL2398991 0.82 ITK (0.57) LCKKDRSSTR5ITKAURKB
SCHEMBL2398982 0.82 ITK (0.57) LCKKDRSSTR5ITKAURKB
SCHEMBL2369709 0.80 NPC1 (0.52) LCKRAB9ANPC1SMN1; SMN2SSTR5
SCHEMBL10286645 0.79 ITK (0.44) LCKKDRSSTR5ITKAURKB
SCHEMBL2370127 0.78 NPC1 (0.44) LCKRAB9ANPC1SMN1; SMN2SSTR5
SCHEMBL10285818 0.77 NPC1 (0.49) LCKRAB9ANPC1SMN1; SMN2SSTR5
SCHEMBL2370220 0.77 ALDH1A1 (0.59) LCKRAB9ANPC1SMN1; SMN2POLB
SCHEMBL807804 0.75 LCK (0.46) LCKRAB9AKDRNPC1SMN1; SMN2
SCHEMBL807541 0.75 ITK (0.55) LCKSSTR5ITKAURKBRORC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012035055-A1 NOVEL COMPOUNDS GLAXO GROUP LIMITED (GB) 2012-03-22 WO disclosed