SCHEMBL807713

SCHEMBL807713

C[C@@H]1CN(Cc2cc(Nc3nc4cccnc4s3)nc(NCCNC(=O)OC(C)(C)C)n2)C[C@H](C)O1

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ITK Q08881 3/20 0.41
LCK P06239 2/20 0.41
AURKB Q96GD4 2/20 0.41
BRD4 O60885 3/20 0.37
BCHE P06276 1/20 0.37
RORC P51449 1/20 0.36
DHODH Q02127 1/20 0.36
ADORA2A P29274 3/20 0.35
ADORA2B P29275 2/20 0.35
ADORA3 P0DMS8 2/20 0.34
ADORA1 P30542 1/20 0.34
OPRM1 P35372 1/20 0.34
OPRD1 P41143 1/20 0.34
OPRK1 P41145 1/20 0.34
OGFRL1 Q5TC84 1/20 0.34
KDM4E B2RXH2 1/20 0.33
HSD17B10 Q99714 1/20 0.33
NPC1 O15118 1/20 0.33
POLB P06746 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL807917 0.77 LCK (0.39) ITKLCKAURKBRORCDHODH
SCHEMBL179069 0.75 ITK (0.61) ITKLCKAURKB
SCHEMBL807803 0.74 ITK (0.58) ITKLCKAURKBBRD4RORC
SCHEMBL12470060 0.73 LCK (0.47) ITKLCKAURKBRORCDHODH
SCHEMBL141393 0.68 ITK (0.59) ITKLCKAURKBRORCDHODH
SCHEMBL141392 0.68 ITK (0.59) ITKLCKAURKBRORCDHODH
SCHEMBL807802 0.66 NPC1 (0.47) ITKLCKAURKBBRD4NPC1
SCHEMBL807946 0.66 ITK (0.58) ITKLCKAURKBRORCDHODH
SCHEMBL138603 0.66 ITK (0.71) ITKLCKAURKBRORCDHODH
SCHEMBL807540 0.66 ITK (0.46) ITKLCKAURKBRORCDHODH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012035055-A1 NOVEL COMPOUNDS GLAXO GROUP LIMITED (GB) 2012-03-22 WO disclosed