SCHEMBL8078129

SCHEMBL8078129

CC(C)(C)[Si](OC1CC=C(OS(=O)(=O)C(F)(F)F)Cc2ccccc21)(c1ccccc1)c1ccccc1

nearest known ligand 0.37

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 1/20 0.31
DRD1 P21728 1/20 0.31
DRD4 P21917 1/20 0.31
DRD5 P21918 1/20 0.31
DRD3 P35462 1/20 0.31
AKR1C3 P42330 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8078283 0.77 CES2 (0.32)
SCHEMBL25106735 0.76 BACE1 (0.33) DRD2DRD1DRD4DRD5DRD3
SCHEMBL8078069 0.75 ABL1 (0.35)
SCHEMBL8078312 0.75 DRD2 (0.33) DRD2DRD1DRD4DRD5DRD3
SCHEMBL8078315 0.75
SCHEMBL7720307 0.71 DRD2 (0.35) DRD2DRD1DRD4DRD5DRD3
SCHEMBL25380914 0.69 SMYD2 (0.36)
SCHEMBL537975 0.68 CA2 (0.33) DRD2DRD4DRD3
SCHEMBL18149472 0.68 SMYD2 (0.31)
SCHEMBL3519412 0.67 DRD2 (0.33) DRD2DRD1DRD4DRD5DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1030834-A1 BENZOCYCLOHEPTENE DERIVATIVES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-08-30 EP disclosed
WO-1999024397-A1 BENZOCYCLOHEPTENE DERIVATIVES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1999-05-20 WO disclosed