SCHEMBL8078434

SCHEMBL8078434

CC(=O)OCc1ccc(CBr)cc1OCOCC[Si](C)(C)C

nearest known ligand 0.37

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.37
TSHR P16473 1/20 0.32
ALDH1A1 P00352 1/20 0.32
CYP4F2 P78329 1/20 0.31
CYP4A11 Q02928 1/20 0.31
MAPT P10636 1/20 0.31
HPGD P15428 1/20 0.31
ALOX5AP P20292 1/20 0.30
FEN1 P39748 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1467378 0.72 CYP3A4 (0.46) CYP3A4TSHRALDH1A1CYP4F2CYP4A11
SCHEMBL4050696 0.70 TP53 (0.33) ALOX5APFEN1
SCHEMBL336664 0.69 CYP4F2 (0.49) CYP3A4TSHRALDH1A1CYP4F2CYP4A11
SCHEMBL4050421 0.68 CYP19A1 (0.40) CYP3A4TSHRALDH1A1MAPTHPGD
SCHEMBL23580858 0.68 NPC1 (0.41) CYP4F2CYP4A11HPGDALOX5APFEN1
SCHEMBL6042263 0.68 PDE10A (0.35) TSHRALDH1A1MAPTHPGDALOX5AP
SCHEMBL5432902 0.67 BCHE (0.38) TSHRALDH1A1CYP4F2CYP4A11
SCHEMBL6581703 0.67 CA5A (0.52) CYP3A4TSHRALDH1A1
SCHEMBL7083354 0.66 KDM4E (0.52) ALDH1A1HPGD
SCHEMBL8950532 0.66 DRD2 (0.47) CYP3A4ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6153641-A Pharmaceutically active compounds ASTRA AKTIEBOLAG (SE) 2000-11-28 US disclosed
EP-0925296-A1 NEW PHARMACEUTICALLY ACTIVE COMPOUNDS Astra Aktiebolag (SE) 1999-06-30 EP disclosed
WO-1998011102-A1 NEW PHARMACEUTICALLY ACTIVE COMPOUNDS ASTRA AKTIEBOLAG (SE) 1998-03-19 WO disclosed