SCHEMBL8079176

SCHEMBL8079176

COC(=O)Oc1[nH]nc(C#N)c1C

nearest known ligand 0.32

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 1/20 0.32
ALDH1A1 P00352 1/20 0.31
GAA P10253 1/20 0.31
HPGD P15428 1/20 0.31
EPHX2 P34913 1/20 0.30
PLCG1 P19174 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8090562 0.82 GAA (0.34) LRRK2GAAEPHX2
SCHEMBL7104339 0.78 DYRK1A (0.37) ALDH1A1GAAHPGD
SCHEMBL8086319 0.71 LRRK2 (0.32) LRRK2ALDH1A1GAAHPGD
SCHEMBL22890673 0.66 HSD17B10 (0.48) ALDH1A1GAAHPGD
SCHEMBL12000340 0.64
SCHEMBL15554853 0.64
SCHEMBL11262568 0.62 KDM4E (0.32) ALDH1A1HPGD
SCHEMBL12050434 0.60 EPHX2 (0.33) EPHX2
SCHEMBL11112731 0.60 KDM4E (0.33) ALDH1A1HPGD
SCHEMBL7765129 0.59 HCAR2 (0.44) GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1051431-A1 THROMBIN INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 2000-11-15 EP disclosed
WO-1999037668-A1 THROMBIN INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 1999-07-29 WO disclosed