SCHEMBL8079309

SCHEMBL8079309

CCC(O)(O)OC(=O)c1ccc(N)cc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 4/20 0.58
LMNA P02545 3/20 0.58
CYP3A4 P08684 3/20 0.58
MAOA P21397 2/20 0.58
TSHR P16473 2/20 0.51
CYP2C19 P33261 2/20 0.51
CYP2C9 P11712 1/20 0.51
PDE4D Q08499 1/20 0.51
NPC1 O15118 3/20 0.49
RAB9A P51151 3/20 0.49
MAPT P10636 2/20 0.49
ALDH1A1 P00352 1/20 0.49
CYP2D6 P10635 3/20 0.47
HTR3A P46098 1/20 0.47
HRH3 Q9Y5N1 1/20 0.47
BLM P54132 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
PHLPP2 Q6ZVD8 1/20 0.46
SCN1A P35498 2/20 0.44
SCN2A Q99250 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2788007 0.91 CYP1A2 (0.45) CYP1A2LMNACYP3A4MAOATSHR
SCHEMBL2788009 0.84 ALDH1A1 (0.52) CYP1A2TSHRCYP2C19MAPTALDH1A1
SCHEMBL23486834 0.82 CYP1A2 (0.58) CYP1A2LMNACYP3A4MAOATSHR
SCHEMBL3162941 0.81 CYP2D6 (0.57) CYP1A2LMNATSHRCYP2C19NPC1
SCHEMBL27611708 0.79 CYP1A2 (0.54) CYP1A2LMNACYP3A4MAOATSHR
SCHEMBL2064890 0.79 CYP1A2 (0.50) CYP1A2LMNACYP3A4MAOATSHR
SCHEMBL380152 0.77 CA12 (0.57) CYP1A2LMNACYP3A4MAOATSHR
SCHEMBL2064891 0.77 CYP1A2 (0.51) CYP1A2LMNACYP3A4MAOATSHR
SCHEMBL11640194 0.77 CYP1A2 (0.51) CYP1A2LMNACYP3A4MAOATSHR
SCHEMBL13492201 0.76 LMNA (0.50) CYP1A2LMNACYP3A4MAOATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6120757-A COSMETICS; THERAPY FOR SKIN DISORDERS, HAIR SOCIETE L'OREAL S.A. (FR) 2000-09-19 US disclosed