SCHEMBL8080052

SCHEMBL8080052

O=C(O)c1c2ccccc2nc2c(C(=O)O)cccc12

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.64
NR4A1 P22736 1/20 0.52
NR4A2 P43354 1/20 0.52
NR4A3 Q92570 1/20 0.52
PDE10A Q9Y233 4/20 0.51
CDC25B P30305 1/20 0.50
DHODH Q02127 5/20 0.49
LMNA P02545 2/20 0.49
TSHR P16473 1/20 0.47
KDM4E B2RXH2 3/20 0.47
MEN1 O00255 3/20 0.47
KMT2A Q03164 3/20 0.47
CYP2C19 P33261 2/20 0.47
HSD17B10 Q99714 2/20 0.47
CYP1A2 P05177 1/20 0.47
GLA P06280 1/20 0.47
HPGD P15428 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.46
CASP1 P29466 1/20 0.44
CASP7 P55210 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21119051 0.83 ALDH1A1 (0.64) ALDH1A1NR4A1NR4A2NR4A3PDE10A
SCHEMBL13313361 0.83 CYP1A2 (0.60) ALDH1A1PDE10ADHODHLMNATSHR
SCHEMBL9330496 0.81 PDE10A (0.58) ALDH1A1PDE10ADHODHLMNATSHR
SCHEMBL641899 0.81 PDE10A (0.66) ALDH1A1PDE10ADHODHLMNATSHR
SCHEMBL29377848 0.81 PDE10A (0.66) ALDH1A1PDE10ADHODHLMNATSHR
SCHEMBL7028209 0.79 KMT2A (0.52) ALDH1A1NR4A1NR4A2NR4A3PDE10A
Iodide SCHEMBL8029601 0.79 PDE10A (0.63) ALDH1A1PDE10ADHODHLMNATSHR
Hydrochloric Acid SCHEMBL9597551 0.79 PDE10A (0.63) ALDH1A1PDE10ADHODHLMNATSHR
Iodide SCHEMBL8029606 0.79 PDE10A (0.63) ALDH1A1PDE10ADHODHLMNATSHR
SCHEMBL68995 0.79 ALDH1A1 (0.88) ALDH1A1NR4A1NR4A2NR4A3DHODH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5939568-A Accelerated catalysis of olefinic epoxidations THE SCRIPPS RESEARCH INSTITUTE (US) 1999-08-17 US claimed
WO-1998033786-A9 ACCELERATED CATALYSIS OF OLEFINIC EPOXIDATIONS 1998-12-30 WO claimed
WO-1998033786-A1 ACCELERATED CATALYSIS OF OLEFINIC EPOXIDATIONS THE SCRIPPS RESEARCH INSTITUTE (US) 1998-08-06 WO claimed
EP-0904434-B1 ACID-DYEABLE FIBRE DSM NV (NL) 2000-09-20 EP disclosed
US-6074749-A POLYAMIDE HAVING AN AMINO END GROUP CONTENT OF LESS THAN 10 MEQ/KG DSM N.V. (NL) 2000-06-13 US disclosed
US-5939568-A Accelerated catalysis of olefinic epoxidations THE SCRIPPS RESEARCH INSTITUTE (US) 1999-08-17 US disclosed
EP-0904434-A1 ACID-DYEABLE FIBRE DSM N.V. (NL) 1999-03-31 EP disclosed
WO-1998033786-A9 ACCELERATED CATALYSIS OF OLEFINIC EPOXIDATIONS 1998-12-30 WO disclosed
WO-1998033786-A1 ACCELERATED CATALYSIS OF OLEFINIC EPOXIDATIONS THE SCRIPPS RESEARCH INSTITUTE (US) 1998-08-06 WO disclosed
WO-1997046746-A1 ACID-DYEABLE FIBRE DSM N.V. (NL) 1997-12-11 WO disclosed