SCHEMBL8080356

SCHEMBL8080356

Nc1cc(Cl)ccc1C(=O)c1cccc(O)c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C4 P17516 1/20 0.49
AKR1C3 P42330 1/20 0.49
AKR1C2 P52895 1/20 0.49
AKR1C1 Q04828 1/20 0.49
ABL1 P00519 1/20 0.47
PARP1 P09874 1/20 0.47
FASN P49327 1/20 0.46
ALOX15 P16050 2/20 0.46
ALDH1A1 P00352 2/20 0.46
HPGD P15428 1/20 0.46
ALOX12 P18054 1/20 0.46
MAPK1 P28482 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
HSD17B10 Q99714 1/20 0.46
MAPT P10636 2/20 0.45
CLK1 P49759 1/20 0.45
DYRK1A Q13627 1/20 0.45
DYRK1B Q9Y463 1/20 0.45
HSD17B1 P14061 3/20 0.44
HSD17B2 P37059 3/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4851741 0.89 RECQL (0.55) AKR1C4AKR1C3AKR1C2AKR1C1PARP1
SCHEMBL19774168 0.84 MEN1 (0.57) AKR1C4AKR1C3AKR1C2AKR1C1PARP1
SCHEMBL1041696 0.83 MAPT (0.61) ABL1ALOX15ALDH1A1MAPTTDP1
SCHEMBL31366555 0.83 MAPT (0.61) ABL1ALOX15ALDH1A1MAPTTDP1
SCHEMBL8956721 0.83 PARP1 (0.49) ABL1PARP1ALOX15ALDH1A1SMN1; SMN2
SCHEMBL2241001 0.82 MAPK1 (0.58) ABL1ALOX15ALDH1A1HPGDALOX12
SCHEMBL8080314 0.80 MAPT (0.67) PARP1FASNALDH1A1MAPTCLK1
SCHEMBL5618019 0.80 RAB9A (0.55) ABL1PARP1ALDH1A1HPGDMAPK1
SCHEMBL11392123 0.78 TSHR (0.61) AKR1C4AKR1C3AKR1C2AKR1C1PARP1
SCHEMBL8956523 0.77 ALOX15 (0.50) PARP1ALOX15ALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6100254-A Inhibitors of protein tyrosine kinases BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 2000-08-08 US disclosed
WO-1999019306-A2 2,3-BENZODIAZEPIN-2-ONE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS INHIBITORS OF PROTEIN TYROSINE KINASES BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 1999-04-22 WO disclosed