SCHEMBL8081656

SCHEMBL8081656

CCc1cc2c(cc1Br)C(C)(C)CCO2

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
RXRA P19793 5/20 0.42
HNF4A P41235 1/20 0.42
RARA P10276 4/20 0.39
RARB P10826 4/20 0.39
RARG P13631 4/20 0.39
MAP3K14 Q99558 2/20 0.38
CYP26A1 O43174 1/20 0.37
CYP26B1 Q9NR63 1/20 0.37
KDM4E B2RXH2 1/20 0.30
PTGS1 P23219 1/20 0.30
PTGS2 P35354 1/20 0.30
SSTR5 P35346 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9009683 0.80 RARA (0.34) RXRAHNF4ARARARARBRARG
SCHEMBL8089804 0.79 RXRA (0.38) RXRAHNF4ARARARARBRARG
SCHEMBL8081756 0.79 RARA (0.38) RXRAHNF4ARARARARBRARG
SCHEMBL14376650 0.78 RXRA (0.46) RXRAHNF4ARARARARBRARG
SCHEMBL9850251 0.78 RXRA (0.56) RXRAHNF4ARARARARBRARG
SCHEMBL6668058 0.78 RXRA (0.50) RXRAHNF4ARARARARBRARG
SCHEMBL9850143 0.72 RXRA (0.53) RXRAHNF4ARARARARBRARG
SCHEMBL6668009 0.72 RXRA (0.47) RXRAHNF4ARARARARBRARG
SCHEMBL6669631 0.71 MAP3K14 (0.43) RXRAHNF4ARARARARBRARG
SCHEMBL30250112 0.70 LMNA (0.46) RXRAHNF4ARARARARBRARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0740665-B1 PROCESS FOR PREPARING 4,4-DIALKYL-6-HALO-CHROMANS OR THIOCHROMANS USEFUL AS PHARMACEUTICAL INTERMEDIATES ALLERGAN SALES INC (US) 2000-12-06 EP disclosed
US-5519150-A Process for preparing 4,4-dialkyl-6-halo-chromans or thiochromans useful as pharmaceutical intermediates ALLERGAN (US) 1996-05-21 US disclosed
US-5420295-A Process for preparing 4,4-dialkyl-6-halo-chromans or thiochromans useful as pharmaceutical intermediates ALLERGAN, INC. (US) 1995-05-30 US disclosed