SCHEMBL8082005

SCHEMBL8082005

Nc1cc(C2(S(=O)(=O)c3cc(F)cc(F)c3)CC2)nc(-c2ccc(NC(=O)NCCO)cc2)n1

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 7/20 0.41
MTOR P42345 5/20 0.41
NAMPT P43490 8/20 0.39
PIK3CD O00329 7/20 0.39
PIK3CB P42338 1/20 0.39
PIK3CG P48736 1/20 0.39
CA12 O43570 1/20 0.37
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
CA4 P22748 1/20 0.37
CA7 P43166 1/20 0.37
CA9 Q16790 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8091160 0.95 NAMPT (0.38) PIK3CAMTORNAMPTPIK3CDPIK3CB
SCHEMBL8089000 0.92 PIK3CD (0.40) PIK3CAMTORNAMPTPIK3CDCA12
SCHEMBL8100146 0.90 CA1 (0.41) PIK3CAMTORNAMPTPIK3CDPIK3CB
SCHEMBL8093138 0.90 NAMPT (0.40) PIK3CAMTORNAMPTPIK3CDPIK3CB
SCHEMBL8090241 0.89 NAMPT (0.43) PIK3CAMTORNAMPTPIK3CDPIK3CB
SCHEMBL8090391 0.88 CA1 (0.41) PIK3CAMTORNAMPTPIK3CDCA12
SCHEMBL8104051 0.88 NAMPT (0.38) PIK3CAMTORNAMPTPIK3CD
SCHEMBL8098775 0.88 CA1 (0.43) PIK3CAMTORNAMPTPIK3CDPIK3CB
SCHEMBL8089917 0.87 PIK3CA (0.39) PIK3CAMTORNAMPTPIK3CDPIK3CG
SCHEMBL8093959 0.87 PIK3CA (0.38) PIK3CAMTORNAMPTPIK3CDPIK3CB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009007748-A2 TRISUBSTITUTED PYRIMIDINE DERIVATIVES FOR THE TREATMENT OF PROLIFERATIVE DISEASES ASTRAZENECA AB (SE) 2009-01-15 WO disclosed