SCHEMBL8083085

SCHEMBL8083085

O=C(CBr)NC(c1ccccc1)(c1ccccc1)c1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 2/20 0.42
GSK3B P49841 2/20 0.42
KCNN4 O15554 3/20 0.41
CYP1A2 P05177 2/20 0.39
CYP3A4 P08684 2/20 0.39
RECQL P46063 1/20 0.39
KIF11 P52732 1/20 0.38
CYP2C19 P33261 1/20 0.38
HIF1A Q16665 1/20 0.38
HDAC3 O15379 3/20 0.38
HDAC4 P56524 3/20 0.38
HDAC1 Q13547 3/20 0.38
HDAC7 Q8WUI4 3/20 0.38
HDAC2 Q92769 3/20 0.38
HDAC10 Q969S8 3/20 0.38
HDAC11 Q96DB2 3/20 0.38
HDAC8 Q9BY41 3/20 0.38
HDAC6 Q9UBN7 3/20 0.38
HDAC9 Q9UKV0 3/20 0.38
HDAC5 Q9UQL6 3/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7923982 0.80 KCNN4 (0.41) KCNN4CYP1A2CYP3A4RECQLKIF11
SCHEMBL27548806 0.80 KCNN4 (0.41) PTPN1KCNN4CYP1A2CYP3A4RECQL
SCHEMBL28777735 0.80 KCNN4 (0.41) KCNN4CYP1A2CYP3A4RECQLKIF11
SCHEMBL12914773 0.80 KCNN4 (0.50) KCNN4CYP1A2CYP3A4RECQLCYP2C19
SCHEMBL31370489 0.80 CYP1A2 (0.58) KCNN4CYP1A2CYP3A4RECQLKIF11
SCHEMBL28769203 0.78 CYP1A2 (0.41) PTPN1KCNN4CYP1A2CYP3A4RECQL
SCHEMBL27538108 0.78 KCNN4 (0.39) PTPN1KCNN4CYP1A2CYP3A4RECQL
SCHEMBL30564476 0.78 KIF11 (0.50) KCNN4CYP1A2CYP3A4RECQLKIF11
SCHEMBL29872151 0.78 L3MBTL1 (0.49) CYP1A2CYP2C19HIF1AKDM4EMEN1
SCHEMBL12286073 0.77 ALOX5 (0.51) KCNN4CYP3A4RECQLCYP2C19MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0757982-B1 Biphenylic compounds, process for their preparations and intermediates for this process, their use as 5-alpha-reductase inhibitors and pharmaceutical compositions containing them HOECHST MARION ROUSSEL INC (FR) 2000-09-20 EP disclosed
US-5965763-A Biphenyl compounds HOECHST MARION ROUSSEL (FR) 1999-10-12 US disclosed
US-5827887-A 5-ALPHA REDUCTASE INHIBITORS ROUSSEL UCLAF (FR) 1998-10-27 US disclosed
EP-0757982-A1 Biphenylic compounds, process for their preparations and intermediates for this process, their use as 5-alpha-reductase inhibitors and pharmaceutical compositions containing them ROUSSEL UCLAF (FR) 1997-02-12 EP disclosed