SCHEMBL8083399

SCHEMBL8083399

OCCN(CCO)CCCCc1ccccc1

nearest known ligand 0.70

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.56
SIGMAR1 Q99720 3/20 0.55
CHRM2 P08172 1/20 0.55
HTR1A P08908 1/20 0.55
ADRA2A P08913 1/20 0.55
CHRM1 P11229 1/20 0.55
DRD1 P21728 1/20 0.55
SLC6A2 P23975 1/20 0.55
SLC6A4 P31645 1/20 0.55
ADRA1A P35348 1/20 0.55
OPRM1 P35372 1/20 0.55
DRD3 P35462 1/20 0.55
SLC6A3 Q01959 1/20 0.55
TDP1 Q9NUW8 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6056146 0.98 KCNH2 (0.59) KCNH2SIGMAR1CHRM2HTR1AADRA2A
SCHEMBL8086575 0.98 KCNH2 (0.59) KCNH2SIGMAR1CHRM2HTR1AADRA2A
Hydrochloric Acid SCHEMBL3028479 0.96 KCNH2 (0.57) KCNH2SIGMAR1CHRM2HTR1AADRA2A
SCHEMBL1299303 0.94 CHRM2 (0.62) KCNH2SIGMAR1CHRM2HTR1AADRA2A
SCHEMBL6706300 0.89 KCNH2 (0.66) KCNH2SIGMAR1CHRM2HTR1AADRA2A
SCHEMBL11699577 0.87 SIGMAR1 (0.69) KCNH2SIGMAR1CHRM2HTR1AADRA2A
SCHEMBL10662405 0.87 SIGMAR1 (0.69) KCNH2SIGMAR1CHRM2HTR1AADRA2A
Trolamine SCHEMBL671041 0.85 KCNH2 (0.68) KCNH2SIGMAR1CHRM2HTR1AADRA2A
Trolamine SCHEMBL11590482 0.85 KCNH2 (0.68) KCNH2SIGMAR1CHRM2HTR1AADRA2A
SCHEMBL6567560 0.85 OPRK1 (0.60) OPRM1DRD3TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0711763-B1 1,4-DI(PHENYLALKYL)PIPERAZINE DERIVATIVES SANTEN PHARMACEUTICAL CO LTD (JP) 2000-10-18 EP disclosed
US-5736546-A BRAIN DISORDERS; PSYCHOLOGICAL DISORDERS SANTEN PHARMACEUTICAL CO., LTD. (JP) 1998-04-07 US disclosed
EP-0711763-A1 NOVEL 1,4-DI(PHENYLALKYL)PIPERAZINE DERIVATIVE SANTEN PHARMACEUTICAL CO., LTD. (JP) 1996-05-15 EP disclosed