SCHEMBL8083712

SCHEMBL8083712

CCCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC(c1ccccc1)c1ccccc1

nearest known ligand 0.67

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CTSK P43235 16/20 0.67
CTSS P25774 4/20 0.59
HDAC4 P56524 1/20 0.50
HDAC1 Q13547 1/20 0.50
REN P00797 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26436628 0.89 CTSK (0.79) CTSKCTSS
SCHEMBL7367960 0.89 CTSK (0.60) CTSKCTSSHDAC4HDAC1REN
SCHEMBL26436627 0.88 CTSK (0.64) CTSKCTSSHDAC4HDAC1REN
SCHEMBL8088476 0.87 CTSK (0.56) CTSKCTSS
SCHEMBL26436630 0.87 CTSK (0.63) CTSKCTSSHDAC4HDAC1REN
SCHEMBL26436631 0.87 CTSK (0.66) CTSKCTSSREN
SCHEMBL25492163 0.87 NPSR1 (0.58) CTSKCTSSHDAC4HDAC1
SCHEMBL22479132 0.84 CTSK (0.50) CTSKCTSSHDAC4HDAC1REN
SCHEMBL22527176 0.84 CTSK (0.50) CTSKCTSSHDAC4HDAC1REN
SCHEMBL23454631 0.84 HDAC4 (0.65) CTSKCTSSHDAC4HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1041064-A2 N-substituted alpha aminoacid amides as calcium channel modulators ELI LILLY AND COMPANY LIMITED (GB) 2000-10-04 EP disclosed