SCHEMBL8084023

SCHEMBL8084023

COC(=O)/C(=C(\C)c1ccc(S(C)(=O)=O)cc1)c1ccc(F)cc1

nearest known ligand 0.58

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
FAAH O00519 1/20 0.48
MGLL Q99685 1/20 0.48
PTGS2 P35354 5/20 0.48
AKR1C2 P52895 1/20 0.47
AKR1C1 Q04828 1/20 0.47
AKR1C3 P42330 1/20 0.47
F2 P00734 1/20 0.46
PRSS1 P07477 1/20 0.46
PRSS2 P07478 1/20 0.46
PRSS3 P35030 1/20 0.46
EPHX2 P34913 2/20 0.45
ESR2 Q92731 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5336468 0.87 PTGS2 (0.60) FAAHMGLLPTGS2AKR1C2AKR1C1
SCHEMBL5336464 0.87 PTGS2 (0.60) FAAHMGLLPTGS2AKR1C2AKR1C1
SCHEMBL5336461 0.87 PTGS2 (0.60) FAAHMGLLPTGS2AKR1C2AKR1C1
SCHEMBL8092899 0.84 PTGS2 (0.57) FAAHMGLLPTGS2AKR1C2AKR1C1
SCHEMBL7844135 0.75 PTGS2 (0.57) FAAHMGLLPTGS2AKR1C2AKR1C1
SCHEMBL4030635 0.74 PTGS2 (0.62) PTGS2AKR1C2AKR1C1AKR1C3ESR2
SCHEMBL6050635 0.74 CES2 (0.64) FAAHMGLLPTGS2AKR1C2AKR1C1
SCHEMBL7880898 0.74 PTGS2 (0.50) FAAHMGLLPTGS2AKR1C2AKR1C1
SCHEMBL7829898 0.74 PTGS2 (0.50) FAAHMGLLPTGS2AKR1C2AKR1C1
SCHEMBL8125071 0.74 PTGS2 (0.50) FAAHMGLLPTGS2AKR1C2AKR1C1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0882015-B1 DIPHENYL STILBENES AS PRODRUGS TO COX-2 INHIBITORS MERCK FROSST CANADA INC (CA) 2000-12-27 EP claimed
US-5733909-A ANTIINFLAMMATORY AGENTS; ANALGESICS; ANTIPYRETIC AGENT MERCK FROSST CANADA, INC. (CA) 1998-03-31 US claimed
EP-0882015-B1 DIPHENYL STILBENES AS PRODRUGS TO COX-2 INHIBITORS MERCK FROSST CANADA INC (CA) 2000-12-27 EP disclosed
US-5733909-A ANTIINFLAMMATORY AGENTS; ANALGESICS; ANTIPYRETIC AGENT MERCK FROSST CANADA, INC. (CA) 1998-03-31 US disclosed