SCHEMBL8084366

SCHEMBL8084366

CC(=O)Nc1cc(Cl)c(=O)n(C2c3cc(C#N)ccc3OC(C)(C)C2O)c1

nearest known ligand 0.54

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ABCC9 O60706 15/20 0.54
ABCC8 Q09428 2/20 0.51
KCNJ11 Q14654 2/20 0.51
KCNJ8 Q15842 2/20 0.51
CYP1A2 P05177 1/20 0.51
CYP2D6 P10635 1/20 0.51
CYP2C9 P11712 1/20 0.51
CYP2C19 P33261 1/20 0.51
LMNA P02545 1/20 0.51
ABCB1 P08183 1/20 0.50
KDM4E B2RXH2 1/20 0.48
DRD2 P14416 1/20 0.47
DRD3 P35462 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8236626 0.89 DRD2 (0.47) ABCC9ABCC8KCNJ11KCNJ8CYP1A2
SCHEMBL8085140 0.89 ABCC9 (0.52) ABCC9ABCC8KCNJ11KCNJ8CYP1A2
SCHEMBL8084958 0.87 ABCC9 (0.54) ABCC9ABCC8KCNJ11KCNJ8CYP1A2
SCHEMBL8085325 0.86 ABCC9 (0.57) ABCC9ABCC8KCNJ11KCNJ8CYP1A2
SCHEMBL8077320 0.86 ABCC9 (0.62) ABCC9ABCC8KCNJ11KCNJ8CYP1A2
SCHEMBL8077163 0.84 ABCC9 (0.58) ABCC9ABCC8KCNJ11KCNJ8CYP1A2
SCHEMBL8084258 0.84 ABCC9 (0.44) ABCC9LMNA
SCHEMBL8085315 0.83 DRD2 (0.44) ABCC9ABCB1KDM4EDRD2DRD3
SCHEMBL8090533 0.83 ABCC9 (0.52) ABCC9ABCC8KCNJ11KCNJ8CYP1A2
SCHEMBL8088422 0.81 ABCC9 (0.60) ABCC9ABCC8KCNJ11KCNJ8CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6153627-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-11-28 US disclosed