SCHEMBL8085012

SCHEMBL8085012

CCCCCOc1c(OC)ccc2c1CCN(C(=O)Cc1ccc(N)cc1)C2

nearest known ligand 0.52

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 6/20 0.52
KMT2A Q03164 2/20 0.46
NPC1 O15118 2/20 0.46
ABCB1 P08183 2/20 0.46
ABCC1 P33527 1/20 0.46
SMN1; SMN2 Q16637 2/20 0.40
ACACB O00763 1/20 0.39
MAPT P10636 1/20 0.39
HPGD P15428 1/20 0.39
HTT P42858 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
DRD2 P14416 1/20 0.38
DRD1 P21728 1/20 0.38
DRD3 P35462 1/20 0.38
RAB9A P51151 1/20 0.38
PTGDR2 Q9Y5Y4 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8085937 0.87 CNR2 (0.43) CNR2KMT2ANPC1ABCB1ABCC1
SCHEMBL23315583 0.78 NPC1 (0.62) KMT2ANPC1ABCB1ABCC1ACACB
SCHEMBL5452259 0.72 MAPT (0.46) KMT2ANPC1ABCB1ABCC1SMN1; SMN2
SCHEMBL4416570 0.72 CNR2 (0.58) CNR2
SCHEMBL11389038 0.71 KMT2A (0.67) KMT2ANPC1ABCB1ABCC1SMN1; SMN2
Ammonia Solution, Strong SCHEMBL5452545 0.71 MAPT (0.46) KMT2ANPC1ABCB1ABCC1SMN1; SMN2
SCHEMBL4418089 0.70 CNR2 (0.82) CNR2KMT2AABCB1MAPTHTT
SCHEMBL6968803 0.70 KMT2A (0.58) KMT2ANPC1ABCB1ABCC1SMN1; SMN2
SCHEMBL4414117 0.69 CNR2 (0.55) CNR2KMT2ANPC1ABCB1SMN1; SMN2
SCHEMBL5132181 0.69 AGTR2 (0.68) KMT2ANPC1ACACBPTGDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6017919-A Compounds and pharmaceutical use thereof JAPAN TOBACCO INC. (JP) 2000-01-25 US disclosed
EP-0887340-A1 NOVEL COMPOUNDS AND PHARMACEUTICAL USE THEREOF Japan Tobacco Inc. (JP) 1998-12-30 EP disclosed