SCHEMBL23315583

SCHEMBL23315583

COc1ccc2c(c1OCc1ccccc1)CCN(C(=O)Cc1ccccc1)C2

nearest known ligand 0.62

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.62
KMT2A Q03164 1/20 0.62
AGTR2 P50052 12/20 0.53
AGTR1 P30556 2/20 0.52
ABCB1 P08183 1/20 0.47
ABCC1 P33527 1/20 0.47
ACACB O00763 1/20 0.47
PTGDR2 Q9Y5Y4 1/20 0.47
GPR183 P32249 1/20 0.47
KDM4E B2RXH2 1/20 0.46
ALOX15 P16050 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5132181 0.89 AGTR2 (0.68) NPC1KMT2AAGTR2AGTR1ACACB
SCHEMBL11747939 0.89 AGTR2 (0.53) NPC1KMT2AAGTR2AGTR1ACACB
SCHEMBL23315440 0.86 KMT2A (0.51) NPC1KMT2AAGTR2ACACBPTGDR2
SCHEMBL21796225 0.85 AGTR2 (0.66) AGTR2AGTR1ACACBKDM4E
SCHEMBL16039389 0.85 AGTR2 (0.52) AGTR2AGTR1ACACBPTGDR2GPR183
SCHEMBL23315308 0.83 KMT2A (0.51) NPC1KMT2APTGDR2ALOX15
SCHEMBL17607347 0.82 ACACB (0.49) NPC1KMT2AAGTR2AGTR1ACACB
SCHEMBL3531595 0.81 AGTR2 (0.68) NPC1KMT2AAGTR2AGTR1GPR183
SCHEMBL11743922 0.80 AGTR2 (0.50) AGTR2AGTR1ACACB
SCHEMBL23315424 0.80 AGTR2 (0.54) AGTR2AGTR1ACACBKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3620454-B1 CARBOXYLIC ACID DERIVATIVE AS AT2R RECEPTOR ANTAGONIST SHANDONG DANHONG PHARMACEUTICAL CO LTD (CN) 2021-05-05 EP disclosed