SCHEMBL8085148

SCHEMBL8085148

COC(=O)c1ccc2c(c1)C(n1cccc(N)c1=O)C(O)C(C)(C)O2

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCC9 O60706 7/20 0.42
KDM4E B2RXH2 3/20 0.38
ALDH1A1 P00352 2/20 0.38
MAPT P10636 2/20 0.38
HPGD P15428 2/20 0.38
NPC1 O15118 2/20 0.38
RAB9A P51151 2/20 0.38
ABCC8 Q09428 2/20 0.37
KCNJ11 Q14654 2/20 0.37
KCNJ8 Q15842 2/20 0.37
CYP1A2 P05177 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
LMNA P02545 1/20 0.37
GLA P06280 1/20 0.36
GAA P10253 1/20 0.36
CASP1 P29466 1/20 0.36
CASP7 P55210 1/20 0.36
ATM Q13315 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8088870 0.85 ABCC9 (0.40) ABCC9KDM4EALDH1A1MAPTHPGD
SCHEMBL7269439 0.85 ABCC9 (0.44) ABCC9ABCC8KCNJ11KCNJ8CYP1A2
SCHEMBL7277059 0.81 KDM4E (0.35) KDM4EALDH1A1MAPTHPGDNPC1
SCHEMBL10697493 0.80 ABCC9 (0.40) ABCC9MAPTRAB9AABCC8KCNJ11
SCHEMBL8077255 0.80 ABCC9 (0.49) ABCC9ABCC8KCNJ11KCNJ8CYP1A2
SCHEMBL7269390 0.80 ABCC9 (0.60) ABCC9KDM4EABCC8KCNJ11KCNJ8
SCHEMBL11395222 0.78 KDM4E (0.48) ABCC9KDM4EALDH1A1MAPTHPGD
SCHEMBL11395215 0.78 KDM4E (0.48) ABCC9KDM4EALDH1A1MAPTHPGD
SCHEMBL11395217 0.78 KDM4E (0.48) ABCC9KDM4EALDH1A1MAPTHPGD
SCHEMBL11399154 0.77 KDM4E (0.50) ABCC9KDM4EALDH1A1MAPTHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6153627-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-11-28 US disclosed
US-6040308-A Chroman derivatives MERCK GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-03-21 US disclosed
US-5387587-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1995-02-07 US disclosed