SCHEMBL8085302

SCHEMBL8085302

CN(C)c1ccc2c(c1)C(n1ccccc1=O)=CC(C)(C)O2

nearest known ligand 0.37

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.37
HPGD P15428 2/20 0.37
HSD17B10 Q99714 2/20 0.37
CYP3A4 P08684 1/20 0.37
HIF1A Q16665 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
CRHBP P24387 1/20 0.32
CRHR2 Q13324 1/20 0.32
MIF P14174 1/20 0.30
BAZ2B Q9UIF8 1/20 0.30
BAZ2A Q9UIF9 1/20 0.30
KDM4E B2RXH2 1/20 0.30
MAPT P10636 1/20 0.30
THRB P10828 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8084219 0.84 KDM4E (0.36) ALDH1A1HPGDHSD17B10CYP3A4CRHBP
SCHEMBL8088499 0.83 TP53 (0.34) CYP3A4TDP1MAPTNPSR1
SCHEMBL8085076 0.83 NPSR1 (0.34) KDM4EMAPTNPSR1MEN1KMT2A
SCHEMBL8077246 0.83 HSD11B1 (0.34) ALDH1A1HPGDTDP1KDM4EMAPT
SCHEMBL8084230 0.83 HRH4 (0.30)
SCHEMBL9796819 0.83 HRH4 (0.34) ALDH1A1HPGDCYP3A4TDP1NPSR1
SCHEMBL8084378 0.82 ATM (0.32) ALDH1A1HPGDMAPT
SCHEMBL7266931 0.81 RXFP1 (0.32) ALDH1A1HSD17B10TDP1
SCHEMBL8085319 0.81 PPIB (0.44) ALDH1A1HPGDHSD17B10TDP1KDM4E
SCHEMBL4260102 0.81 ATM (0.45) HIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6153627-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-11-28 US disclosed
US-6040308-A Chroman derivatives MERCK GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-03-21 US disclosed
US-5387587-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1995-02-07 US disclosed
EP-0273262-A2 Chroman derivatives MERCK PATENT GmbH (DE) 1988-07-06 EP disclosed