SCHEMBL8085869

SCHEMBL8085869

CCCCCOc1cc(C(=O)NC(C)(C)CO)ccc1OC

nearest known ligand 0.68

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
SMPD1 P17405 7/20 0.68
CNR2 P34972 4/20 0.60
PDE4B Q07343 3/20 0.53
PDE4D Q08499 2/20 0.53
PDE4A P27815 1/20 0.53
PDE4C Q08493 1/20 0.53
HDAC3 O15379 1/20 0.51
HDAC2 Q92769 1/20 0.51
TP53 P04637 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28587123 0.81 SMPD1 (1.00) SMPD1CNR2PDE4BPDE4DPDE4A
SCHEMBL28591269 0.81 SMPD1 (1.00) SMPD1CNR2PDE4BPDE4DPDE4A
SCHEMBL4496535 0.79 SMPD1 (0.72) SMPD1PDE4B
SCHEMBL9307263 0.78 SMPD1 (0.76) SMPD1CNR2PDE4B
SCHEMBL9305512 0.78 SMPD1 (0.75) SMPD1PDE4BTP53
SCHEMBL3373445 0.78 SMPD1 (0.71) SMPD1CNR2PDE4B
SCHEMBL28051119 0.78 SMPD1 (0.75) SMPD1PDE4BTP53
SCHEMBL28604170 0.78 SMPD1 (0.75) SMPD1PDE4BTP53
SCHEMBL14452333 0.77 RAB9A (0.50) CNR2HDAC3HDAC2
SCHEMBL1933162 0.77 RAB9A (0.53) SMPD1CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6017919-A Compounds and pharmaceutical use thereof JAPAN TOBACCO INC. (JP) 2000-01-25 US disclosed
EP-0887340-A1 NOVEL COMPOUNDS AND PHARMACEUTICAL USE THEREOF Japan Tobacco Inc. (JP) 1998-12-30 EP disclosed