SCHEMBL8087658

SCHEMBL8087658

N#Cc1cc(CCN)c[nH]1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 4/20 0.41
DRD4 P21917 3/20 0.41
DRD3 P35462 3/20 0.41
HTR1A P08908 2/20 0.41
CCNC P24863 2/20 0.38
CDK8 P49336 2/20 0.38
TAAR1 Q96RJ0 12/20 0.34
HTR2A P28223 3/20 0.34
CYP2A6 P11509 2/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
LOXL2 Q9Y4K0 1/20 0.32
TRPM8 Q7Z2W7 1/20 0.32
DRD1 P21728 3/20 0.31
KDM4E B2RXH2 2/20 0.31
ADRA2A P08913 2/20 0.31
MAPT P10636 2/20 0.31
DRD5 P21918 2/20 0.31
SLC6A2 P23975 2/20 0.31
MAPK1 P28482 2/20 0.31
RECQL P46063 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14493865 0.75
SCHEMBL28873553 0.75
SCHEMBL27952892 0.70
SCHEMBL17410444 0.67
SCHEMBL28110592 0.64 HTR2A (0.46) HTR1ATAAR1HTR2ATRPM8KDM4E
SCHEMBL7221839 0.64 SLC6A4 (0.51) DRD3HTR1ATAAR1HTR2ATRPM8
Hydrochloric Acid SCHEMBL4131221 0.63 TAAR1 (0.37) CCNCCDK8TAAR1
SCHEMBL1225699 0.63 DAO (0.60) DRD2DRD4DRD3HTR1ATAAR1
SCHEMBL3573780 0.63
SCHEMBL18006694 0.63 TRPV4 (0.50) DRD2DRD4DRD3HTR1ATAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1051431-A1 THROMBIN INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 2000-11-15 EP disclosed
EP-0956294-A1 THROMBIN INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 1999-11-17 EP disclosed
WO-1999037668-A1 THROMBIN INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 1999-07-29 WO disclosed
WO-1998006741-A1 THROMBIN INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 1998-02-19 WO disclosed