SCHEMBL28110592

SCHEMBL28110592

COc1cc(CCN)c[nH]1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 6/20 0.46
HTR2C P28335 3/20 0.46
HTR2B P41595 2/20 0.46
KDM4E B2RXH2 1/20 0.44
ATM Q13315 1/20 0.44
TAAR1 Q96RJ0 5/20 0.44
TSHR P16473 3/20 0.42
MAPK1 P28482 1/20 0.42
LMNA P02545 2/20 0.41
CYP1A2 P05177 2/20 0.41
NFKB1 P19838 2/20 0.41
CYP3A4 P08684 1/20 0.41
GLA P06280 1/20 0.41
MAOB P27338 3/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
APEX1 P27695 1/20 0.40
HTR1A P08908 1/20 0.39
MAPT P10636 1/20 0.39
HTR1D P28221 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27952892 0.74
SCHEMBL5154696 0.67
SCHEMBL153674 0.66 TAAR1 (0.64) HTR2AHTR2CHTR2BKDM4EATM
SCHEMBL5173394 0.64
SCHEMBL827905 0.64
SCHEMBL8087658 0.64 DRD2 (0.41) HTR2AKDM4ETAAR1MAPK1LMNA
Hydrochloric Acid SCHEMBL11087070 0.64 TAAR1 (0.62) HTR2AHTR2CHTR2BKDM4EATM
SCHEMBL260789 0.64 GABRA1 (0.45) KDM4EATMLMNACYP1A2CYP3A4
SCHEMBL1225699 0.63 DAO (0.60) HTR2AHTR2CKDM4ETAAR1TSHR
SCHEMBL5171703 0.63

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103664974-B Aryl [a] indole [2,3-g] quinolizine compounds, its preparation method, pharmaceutical composition and application thereof 中国科学院上海药物研究所 2016-12-21 CN disclosed