SCHEMBL8087797

SCHEMBL8087797

CC(=O)Oc1[nH]c2ccccc2c1C

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 2/20 0.63
ADK P55263 2/20 0.63
SLC22A6 Q4U2R8 1/20 0.51
ALDH1A1 P00352 4/20 0.50
HSD17B10 Q99714 3/20 0.50
AHR P35869 1/20 0.50
DAO P14920 1/20 0.50
DDO Q99489 1/20 0.50
HTT P42858 3/20 0.47
MAPT P10636 3/20 0.47
USP2 O75604 2/20 0.47
HPGD P15428 2/20 0.47
KDM4E B2RXH2 2/20 0.46
GAA P10253 2/20 0.46
NR4A2 P43354 2/20 0.46
TP53 P04637 1/20 0.46
KMT2A Q03164 2/20 0.43
ALOX12 P18054 1/20 0.43
PPARG P37231 1/20 0.43
NCOA2 Q15596 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28438445 0.88 GSK3B (0.51) GSK3BADKSLC22A6ALDH1A1HSD17B10
SCHEMBL9264435 0.82 KDM4E (0.49) GSK3BADKALDH1A1HSD17B10DAO
SCHEMBL6471859 0.82 GSK3B (0.59) GSK3BADKSLC22A6ALDH1A1HSD17B10
SCHEMBL28112445 0.81 GSK3B (0.57) GSK3BADKSLC22A6ALDH1A1HSD17B10
SCHEMBL8087793 0.81 GSK3B (0.57) GSK3BADKSLC22A6HSD17B10HTT
SCHEMBL7459854 0.79 KDM4E (0.58) GSK3BADKSLC22A6ALDH1A1HSD17B10
SCHEMBL6526599 0.79 GSK3B (0.56) GSK3BADKSLC22A6ALDH1A1HSD17B10
SCHEMBL11667064 0.77 GSK3B (0.54) GSK3BADKSLC22A6ALDH1A1HSD17B10
SCHEMBL2006899 0.77 AHR (0.57) ALDH1A1HSD17B10AHRDAODDO
SCHEMBL27908888 0.77 KEAP1 (0.47) GSK3BADKALDH1A1HTTMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105308024-A Bicyclic nitrogen-containing aromatic heterocyclic amide compound ASTELLAS PHARMA INC 2016-02-03 CN disclosed
EP-0555537-B1 Endothelin antagonists BANYU PHARMA CO LTD (JP) 2000-11-02 EP disclosed
US-5614498-A OLIGOPEPTIDES, BRONCHDILATORS BANYU PHARMACEUTICAL CO., LTD. (JP) 1997-03-25 US disclosed
US-5496928-A Endothelin antagonistic substance BANYU PHARMACEUTICAL CO., LTD. (JP) 1996-03-05 US disclosed
EP-0555537-A2 Endothelin antagonistic substance BANYU PHARMACEUTICAL CO., LTD. (JP) 1993-08-18 EP disclosed