SCHEMBL8088441

SCHEMBL8088441

CC(Cc1ccc(C#N)cc1)(NC(=O)C1CCCN(Cc2ccccc2Cl)C1)c1cnc[nH]1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.43
KDM4E B2RXH2 1/20 0.43
FNTA P49354 4/20 0.42
FNTB P49356 4/20 0.42
PGGT1B P53609 4/20 0.42
MAPT P10636 2/20 0.41
TP53 P04637 1/20 0.41
CXCR4 P61073 1/20 0.41
AADAT Q8N5Z0 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2C9 P11712 1/20 0.37
GAA P10253 1/20 0.36
HTT P42858 1/20 0.36
ATM Q13315 1/20 0.36
ROCK2 O75116 1/20 0.36
CCR2 P41597 1/20 0.36
ROCK1 Q13464 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8095399 0.93 CYP3A4 (0.44) ALDH1A1KDM4ECYP1A2CYP3A4CYP2C9
SCHEMBL8098292 0.89 ATM (0.38) ALDH1A1KDM4EGAAHTTATM
SCHEMBL8097852 0.88 KDM4E (0.46) ALDH1A1KDM4EFNTAFNTBPGGT1B
SCHEMBL8088938 0.88 KDM4E (0.46) ALDH1A1KDM4EFNTAFNTBPGGT1B
SCHEMBL8103798 0.87 L3MBTL1 (0.39) ALDH1A1KDM4EMAPTTP53CYP1A2
SCHEMBL8101381 0.86 CCR5 (0.38) FNTAFNTBATMCCR2KMT2A
SCHEMBL446561 0.86 ALOX12 (0.40) CCR2KMT2A
SCHEMBL8095905 0.86 GSK3B (0.38) CYP2C9ATMNPSR1
SCHEMBL8088210 0.85 TSHR (0.40) CYP1A2CYP3A4CYP2C9HTTROCK2
SCHEMBL8101586 0.85 GPBAR1 (0.35) MAPTCYP2C9GAANPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6127366-A ANTICARCINOGENIC OR ANTITUMOR AGENTS MERCK & CO., INC. (US) 2000-10-03 US disclosed
US-5817678-A IMIDAZOLE-CONTAINING PIPERIDINE DERIVATIVES, PEPTIDEMIMETIC MERCK & CO., INC. (US) 1998-10-06 US disclosed