SCHEMBL8089127

SCHEMBL8089127

CCOCCNC(=O)CN(CCN(CCN(CC(=O)O)CC(=O)NCCOCC)CC(=O)O)CC(=O)O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BLM P54132 2/20 0.47
PMP22 Q01453 2/20 0.47
TDP1 Q9NUW8 2/20 0.47
KDM4E B2RXH2 1/20 0.47
LMNA P02545 1/20 0.47
CHRM2 P08172 1/20 0.47
ADRA2A P08913 1/20 0.47
ALOX15 P16050 1/20 0.47
TSHR P16473 1/20 0.47
DRD1 P21728 1/20 0.47
SLC6A2 P23975 1/20 0.47
SLC6A4 P31645 1/20 0.47
CYP2C19 P33261 1/20 0.47
ADRA1A P35348 1/20 0.47
DRD3 P35462 1/20 0.47
SLC6A3 Q01959 1/20 0.47
HRH3 Q9Y5N1 1/20 0.47
HSD17B10 Q99714 1/20 0.44
CA1 P00915 15/20 0.44
CA2 P00918 15/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24024217 1.00 BLM (0.47) BLMPMP22TDP1KDM4ELMNA
SCHEMBL24024197 1.00 BLM (0.47) BLMPMP22TDP1KDM4ELMNA
SCHEMBL29344308 0.86 BLM (0.51) BLMPMP22TDP1KDM4ELMNA
SCHEMBL5547592 0.85 BLM (0.50) BLMPMP22TDP1KDM4ELMNA
SCHEMBL14252347 0.85 BLM (0.46) BLMPMP22TDP1KDM4ELMNA
SCHEMBL26261947 0.85 BLM (0.44) BLMPMP22TDP1KDM4ELMNA
SCHEMBL8103783 0.84 TDP1 (0.50) BLMPMP22TDP1KDM4ELMNA
Versetamide SCHEMBL2109367 0.84 TDP1 (0.50) BLMPMP22TDP1KDM4ELMNA
SCHEMBL24024195 0.84 CA1 (0.40) BLMPMP22TDP1KDM4ELMNA
SCHEMBL8877901 0.83 CA1 (0.47) BLMPMP22TDP1KDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0425571-B2 NOVEL MAGNETIC RESONANCE IMAGING AGENTS MALLINCKRODT MEDICAL INC (US) 2000-09-20 EP disclosed
EP-0425571-B1 NOVEL MAGNETIC RESONANCE IMAGING AGENTS MALLINCKRODT INC (US) 1996-09-11 EP disclosed
US-5137711-A PARAMAGNETIC DTPA AND EDTA ALKOXYALKYLAMIDE COMPLEXES AS MRI AGENTS MALLICKRODT MEDICAL, INC. (US) 1992-08-11 US disclosed
US-5130120-A Diethylenetriaminepentaacetic acid or ethylenediamine tetraacetic acid for magnetic resonance imaging MALLINCKRODT MEDICAL, INC. (US) 1992-07-14 US disclosed
EP-0425571-A1 NOVEL MAGNETIC RESONANCE IMAGING AGENTS. MALLINCKRODT INC (US) 1991-05-08 EP disclosed
WO-1990001024-A1 NOVEL MAGNETIC RESONANCE IMAGING AGENTS MALLINCKRODT, INC. (US) 1990-02-08 WO disclosed