SCHEMBL8089248

SCHEMBL8089248

Sc1nccn1-c1ccccn1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.47
TSHR P16473 1/20 0.47
POLB P06746 1/20 0.46
ALDH1A1 P00352 1/20 0.43
HTT P42858 1/20 0.43
HSD17B10 Q99714 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.40
PLD1 Q13393 1/20 0.39
EP300 Q09472 1/20 0.38
KAT2B Q92831 1/20 0.38
RAB9A P51151 1/20 0.37
GRIN2D O15399 1/20 0.36
GRIN3B O60391 1/20 0.36
GRIN1 Q05586 1/20 0.36
GRIN2A Q12879 1/20 0.36
GRIN2B Q13224 1/20 0.36
GRIN2C Q14957 1/20 0.36
GRIN3A Q8TCU5 1/20 0.36
PTK2 Q05397 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27358257 0.76 KDM4E (0.47) KDM4ETSHRPOLBALDH1A1HTT
SCHEMBL8499717 0.76 KDM4E (0.47) KDM4ETSHRPOLBALDH1A1HTT
SCHEMBL17844038 0.76 KDM4E (0.47) KDM4ETSHRPOLBALDH1A1HTT
SCHEMBL353826 0.75 CYP3A4 (0.50) POLBALDH1A1HTTSMN1; SMN2RAB9A
SCHEMBL2269279 0.73 CYP3A4 (0.49) POLBALDH1A1HTTSMN1; SMN2RAB9A
SCHEMBL5594263 0.73 KDR (0.57) KDM4ETSHRPOLB
SCHEMBL9808678 0.73 CCR1 (0.47) KDM4ETSHRALDH1A1SMN1; SMN2RAB9A
SCHEMBL21753738 0.72 KDM4E (0.44) KDM4ETSHRPOLBALDH1A1HTT
SCHEMBL25778550 0.71 KDM4E (0.66) KDM4ETSHRPOLBALDH1A1HTT
SCHEMBL9372056 0.69 TSHR (0.46) KDM4ETSHRPOLBALDH1A1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6043242-A TREATING A MAMMAL AFFLICTED WITH A DISEASE BASED ON HELICOBACTER BACTERIA BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 2000-03-28 US disclosed
EP-0946559-A2 IMIDAZOPYRIDAZINES Byk Gulden Lomberg Chemische Fabrik GmbH (DE) 1999-10-06 EP disclosed
WO-1998028299-A2 IMIDAZOPYRIDAZINES BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 1998-07-02 WO disclosed
EP-0328024-B1 Tetramethylpiperidino-s triazines CIBA GEIGY AG (CH) 1994-12-28 EP disclosed
EP-0249938-B1 Imidazolesulfonamide derivatives, herbicides and a method for inhibiting growth of undesirable plants NISSAN CHEMICAL IND LTD (JP) 1994-12-14 EP disclosed
CN-1020902-C IMIDAZOLE DERIVATIVE AND PROCESSES FOR PREPARING SAME TANAHBE SEIYAKU CO LTD (JP) 1993-05-26 CN disclosed
EP-0270091-B1 IMIDAZOLE DERIVATIVES, PROCESSES FOR THE PREPARATION OF THE SAME, PHARMACEUTICAL COMPOSITIONS COMPRISING THE SAME, THE USE OF THE SAME FOR THE MANUFACTURE OF MEDICAMENTS OF THERAPEUTIC VALUE, AND INTERMEDIATES FORMED DURING SAID PROCESSES TANABE SEIYAKU CO., LTD. (JP) 1992-11-11 EP disclosed
US-5053417-A Antiulcer agents TANABE SEIYAKU CO., LTD. (JP) 1991-10-01 US disclosed
US-5002945-A Antiulcer agents TANABE SEIYAKU CO. LTD. (JP) 1991-03-26 US disclosed
US-4996217-A Antiulcer agents TANABE SEIYAKU COMPANY, LTD. (JP) 1991-02-26 US disclosed
EP-0328024-A1 Tetramethylpiperidino-s triazines CIBA-GEIGY AG (CH) 1989-08-16 EP disclosed
US-4830660-A Imidazolesulfonamide derivatives and herbicides NISSAN CHEMICAL INDUSTRIES, LTD. (JP) 1989-05-16 US disclosed
CN-87108111-A Novel imidazole derivative and preparation method thereof 1988-09-28 CN disclosed
EP-0270091-A1 Imidazole derivatives, processes for the preparation of the same, pharmaceutical compositions comprising the same, the use of the same for the manufacture of medicaments of therapeutic value, and intermediates formed during said processes TANABE SEIYAKU CO., LTD. (JP) 1988-06-08 EP disclosed
EP-0249938-A2 Imidazolesulfonamide derivatives, herbicides and a method for inhibiting growth of undesirable plants NISSAN CHEMICAL INDUSTRIES LTD. (JP) 1987-12-23 EP disclosed