SCHEMBL8089523

SCHEMBL8089523

COc1cc[c]c(-c2ccc3ccccc3c2)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 3/20 0.53
CYP2A6 P11509 1/20 0.53
HSD17B1 P14061 1/20 0.43
HSD17B2 P37059 1/20 0.43
CYP11B2 P19099 5/20 0.42
CYP11B1 P15538 4/20 0.42
CYP3A4 P08684 2/20 0.42
CYP2C9 P11712 2/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2B6 P20813 1/20 0.42
CYP2C19 P33261 1/20 0.42
GSTP1 P09211 2/20 0.41
CYP17A1 P05093 2/20 0.41
CYP19A1 P11511 1/20 0.40
PTGS2 P35354 1/20 0.39
CDK5 Q00535 1/20 0.39
CDK5R1 Q15078 1/20 0.39
NQO2 P16083 1/20 0.39
SLC6A2 P23975 1/20 0.39
SLC6A4 P31645 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10918406 0.83 CYP11B1 (0.44) CYP1A2CYP2A6CYP11B2CYP11B1CYP19A1
SCHEMBL7033071 0.82 CA4 (0.43) CYP1A2CYP2A6CYP11B2CYP11B1CYP3A4
SCHEMBL323109 0.81 DYRK1A (0.49) CYP1A2CYP2A6CYP3A4CYP2C9CYP2D6
SCHEMBL2448879 0.80 ESR1 (0.48) CYP1A2HSD17B1HSD17B2CYP11B2CYP11B1
SCHEMBL459934 0.80 CA12 (0.44) CYP1A2HSD17B1HSD17B2CYP3A4CYP2C9
SCHEMBL28480166 0.80 CYP1A2 (0.53) CYP1A2CYP2A6HSD17B1HSD17B2CYP11B2
SCHEMBL8640563 0.80 KAT6A (0.35) CYP1A2CYP2A6HSD17B1HSD17B2CYP11B2
SCHEMBL6987825 0.79 CYP1A2 (0.50) CYP1A2CYP2A6HSD17B1HSD17B2CYP11B2
SCHEMBL10448704 0.79 CYP2A6 (0.50) CYP1A2CYP2A6HSD17B1HSD17B2CYP11B2
SCHEMBL8531326 0.79 LTA4H (0.53) CYP1A2CYP2A6GSTP1KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1051394-A1 POTASSIUM CHANNEL INHIBITORS Icagen, Inc. (US) 2000-11-15 EP disclosed
WO-1999037607-A1 POTASSIUM CHANNEL INHIBITORS ICAGEN, INC. (US) 1999-07-29 WO disclosed
US-4892887-A ANTITUMOR YALE UNIVERSITY (US) 1990-01-09 US disclosed
US-4684747-A ANTITUMOR, ALKYLATING AGENTS YALE UNIVERSITY (US) 1987-08-04 US disclosed