SCHEMBL8089751

SCHEMBL8089751

CCOC(=O)C1CC=CCC1(CC)C(=O)OCC.O=C1c2cccc3c2C(=O)N13

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 0.34
MEN1 O00255 4/20 0.34
ALDH1A1 P00352 6/20 0.34
KDM4E B2RXH2 2/20 0.34
AGTR1 P30556 1/20 0.34
MAPT P10636 3/20 0.33
HPGD P15428 2/20 0.33
ALOX12 P18054 1/20 0.33
GAA P10253 1/20 0.32
LMNA P02545 2/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
ANPEP P15144 1/20 0.32
DPP4 P27487 1/20 0.32
ATM Q13315 1/20 0.32
PDCD1 Q15116 1/20 0.32
CD274 Q9NZQ7 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28404458 0.71 ADAM17 (0.34) KMT2AMEN1ALDH1A1KDM4EGAA
SCHEMBL3662663 0.62 DPP4 (0.44) KMT2AMEN1ALDH1A1HPGDLMNA
SCHEMBL19412129 0.61
SCHEMBL11278859 0.60 NOS3 (0.40) KMT2AMEN1ALDH1A1KDM4EMAPT
SCHEMBL27689559 0.60 DPP4 (0.44) KMT2AMEN1KDM4EGAALMNA
SCHEMBL9517115 0.60 MAPT (0.33) KMT2AMEN1ALDH1A1KDM4EMAPT
SCHEMBL11018073 0.59 DPP4 (0.60) KMT2AMEN1ALDH1A1KDM4EMAPT
SCHEMBL28405609 0.57 MEN1 (0.33) KMT2AMEN1ALDH1A1KDM4EGAA
SCHEMBL19585730 0.57 ADAM17 (0.57) ALDH1A1L3MBTL1
SCHEMBL28433212 0.57 SMN1; SMN2 (0.53) ALDH1A1GAAL3MBTL1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6018054-A INTERMEDIATE COMPOUNDS FOR PREPARING NOVEL QUINOLONE AND NAPHTHYRIDONE DERIVATIVES WHICH ARE SUBSTITUTED IN THE 7-POSITION BY A PARTIALLY HYDROGENATED ISOINDOLINYL RING, USE AS ANTIBACTERIAL AGENTS AND AS FEED ADDITIVES BAYER AKTIENGESELLSCHAFT (DE) 2000-01-25 US disclosed