SCHEMBL8090075

SCHEMBL8090075

ClC(c1ccccc1)c1nnn[nH]1

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.39
KDM4E B2RXH2 2/20 0.36
ALDH1A1 P00352 2/20 0.36
HPGD P15428 1/20 0.36
KMT2A Q03164 1/20 0.33
ATM Q13315 1/20 0.33
L3MBTL1 Q9Y468 3/20 0.32
SLC6A2 P23975 2/20 0.31
SLC6A4 P31645 2/20 0.31
SLC6A3 Q01959 2/20 0.31
CFTR P13569 1/20 0.31
GOPC Q9HD26 1/20 0.31
GAA P10253 1/20 0.31
DPP4 P27487 2/20 0.30
F2 P00734 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7510243 0.79 KMT2A (0.44) TSHRKDM4EALDH1A1KMT2AATM
SCHEMBL11531757 0.79 KMT2A (0.35) TSHRKDM4EALDH1A1KMT2AATM
SCHEMBL10969072 0.78 TSHR (0.34) TSHRKDM4EKMT2AATM
SCHEMBL9090443 0.76 SMN1; SMN2 (0.46) KDM4EALDH1A1HPGDL3MBTL1
SCHEMBL7679328 0.76 KMT2A (0.41) KDM4EALDH1A1KMT2AATM
SCHEMBL8090152 0.76 KMT2A (0.33) TSHRKDM4EALDH1A1KMT2AATM
SCHEMBL9090435 0.76 CES2 (0.33) TSHRKDM4EALDH1A1KMT2AATM
SCHEMBL9384051 0.76 DPP4 (0.39) KMT2AATMDPP4F2
Hydrochloric Acid SCHEMBL9985742 0.74 DPP4 (0.38) ALDH1A1KMT2AATMDPP4F2
SCHEMBL6470815 0.73 HTR2A (0.34) KDM4EHPGDKMT2AATML3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0829480-B1 Tetrazolyl-substituted quinuclidines as substance P antagonists PFIZER (US) 2000-12-20 EP disclosed
US-5939434-A Tetrazolyl-substituted quinuclidines as substance P antagonists PFIZER PHARMACEUTICALS INC. (JP) 1999-08-17 US disclosed
EP-0829480-A2 Tetrazolyl-substituted quinuclidines as substance P antagonists PFIZER INC. (US) 1998-03-18 EP disclosed