SCHEMBL8090549

SCHEMBL8090549

O=C(O)c1ccc(-c2nnc(-c3ccc(-c4ccc(OCCCOc5ccccc5)cc4)cc3)o2)cc1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 5/20 0.66
RAB9A P51151 5/20 0.66
NR1H4 Q96RI1 1/20 0.64
PKM P14618 1/20 0.60
RARB P10826 5/20 0.55
KDM4E B2RXH2 3/20 0.54
ALDH1A1 P00352 3/20 0.54
TP53 P04637 2/20 0.54
HPGD P15428 2/20 0.54
SMN1; SMN2 Q16637 2/20 0.54
MAPT P10636 3/20 0.53
HSD17B10 Q99714 2/20 0.53
KMT2A Q03164 1/20 0.51
LMNA P02545 1/20 0.50
TSHR P16473 1/20 0.50
PLA2G4B P0C869 1/20 0.50
HDAC6 Q9UBN7 1/20 0.49
PTPN1 P18031 1/20 0.49
CSNK2A2 P19784 1/20 0.48
CSNK2A1 P68400 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7324596 0.97 NPC1 (0.66) NPC1RAB9ANR1H4PKMRARB
SCHEMBL7323297 0.89 RARB (0.70) NPC1RAB9ANR1H4RARBKDM4E
SCHEMBL12171578 0.88 NR1H4 (0.70) NPC1RAB9ANR1H4RARBKDM4E
SCHEMBL7324703 0.87 MAPT (0.64) NPC1RAB9ANR1H4KDM4EALDH1A1
SCHEMBL8086185 0.87 PKM (0.79) RAB9APKMRARBALDH1A1TP53
SCHEMBL7323408 0.87 RARB (0.75) NPC1RAB9ANR1H4RARBKDM4E
SCHEMBL7338309 0.86 NR1H4 (0.68) NPC1RAB9ANR1H4RARBKDM4E
SCHEMBL7314596 0.86 RARB (0.78) NPC1RAB9ANR1H4RARBKDM4E
SCHEMBL8087307 0.86 RARB (0.78) NPC1RAB9ANR1H4RARBKDM4E
SCHEMBL7323524 0.86 NR1H4 (0.64) NPC1RAB9ANR1H4RARBKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1053247-A1 ANTIFUNGAL CYCLOHEXAPEPTIDES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-11-22 EP disclosed
WO-1999040108-A1 NEW COMPOUND FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1999-08-12 WO disclosed