SCHEMBL8090846

SCHEMBL8090846

Nc1cc(C2(S(=O)(=O)c3ccccn3)CCCC2)nc(-c2ccc(NC(=O)NCCO)cc2)n1

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 4/20 0.39
PIK3CA P42336 7/20 0.39
MTOR P42345 3/20 0.39
CHRNA7 P36544 1/20 0.37
CA12 O43570 3/20 0.36
CA1 P00915 3/20 0.36
CA2 P00918 3/20 0.36
CA9 Q16790 3/20 0.36
PIK3CD O00329 8/20 0.36
PIK3CB P42338 1/20 0.36
PIK3CG P48736 1/20 0.36
CNR1 P21554 1/20 0.34
ATR Q13535 1/20 0.34
CA4 P22748 1/20 0.34
CA7 P43166 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8083970 0.98 NAMPT (0.39) NAMPTPIK3CAMTORCHRNA7CA12
SCHEMBL8099754 0.95 CHRNA7 (0.39) NAMPTPIK3CAMTORCHRNA7CA12
SCHEMBL8090849 0.93 NAMPT (0.39) NAMPTPIK3CAMTORCHRNA7CA12
SCHEMBL8098808 0.92 NAMPT (0.39) NAMPTPIK3CAMTORCHRNA7CA12
SCHEMBL8091924 0.89 NAMPT (0.39) NAMPTPIK3CACA12CA1CA2
SCHEMBL8092406 0.88 PIK3CA (0.41) NAMPTPIK3CAMTORCA12CA1
SCHEMBL8090873 0.87 NAMPT (0.38) NAMPTPIK3CACHRNA7CA12CA1
SCHEMBL8098135 0.86 MTOR (0.39) NAMPTPIK3CAMTORPIK3CDPIK3CG
SCHEMBL8084013 0.86 PIK3CA (0.41) NAMPTPIK3CAMTORCA12CA1
SCHEMBL8097518 0.86 KDR (0.38) PIK3CAMTORCA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009007748-A2 TRISUBSTITUTED PYRIMIDINE DERIVATIVES FOR THE TREATMENT OF PROLIFERATIVE DISEASES ASTRAZENECA AB (SE) 2009-01-15 WO disclosed