SCHEMBL8097518

SCHEMBL8097518

Nc1cc(C2(S(=O)(=O)c3ccccn3)CCCC2)nc(-c2ccc(NC(=O)NC3CC3)cc2)n1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 6/20 0.38
EGFR P00533 1/20 0.38
ERBB2 P04626 1/20 0.38
MET P08581 1/20 0.38
MERTK Q12866 1/20 0.38
CA12 O43570 3/20 0.38
CA1 P00915 3/20 0.38
CA2 P00918 3/20 0.38
CA9 Q16790 3/20 0.38
CA4 P22748 2/20 0.38
CA7 P43166 2/20 0.38
KIT P10721 1/20 0.37
FLT3 P36888 1/20 0.37
MAP4K4 O95819 1/20 0.37
EPHX1 P07099 3/20 0.36
RAB9A P51151 2/20 0.36
GAA P10253 1/20 0.36
PIK3CA P42336 2/20 0.36
MTOR P42345 2/20 0.36
EPHX2 P34913 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8090842 0.98 KDR (0.38) KDREGFRERBB2METMERTK
SCHEMBL8091129 0.95 KDR (0.40) KDREGFRERBB2METMERTK
SCHEMBL8084016 0.88 CA12 (0.41) KDRCA12CA1CA2CA9
SCHEMBL8098135 0.87 MTOR (0.39) PIK3CAMTORATR
SCHEMBL8090948 0.86 CA12 (0.41) KDRCA12CA1CA2CA9
SCHEMBL8090849 0.86 NAMPT (0.39) CA12CA1CA2CA9CA4
SCHEMBL8090846 0.86 NAMPT (0.39) CA12CA1CA2CA9CA4
SCHEMBL8096070 0.85 MTOR (0.40) PIK3CAMTORATR
SCHEMBL8092294 0.85 ROCK2 (0.39) CA12CA1CA2CA9PIK3CA
SCHEMBL8099754 0.85 CHRNA7 (0.39) KDRCA12CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009007748-A2 TRISUBSTITUTED PYRIMIDINE DERIVATIVES FOR THE TREATMENT OF PROLIFERATIVE DISEASES ASTRAZENECA AB (SE) 2009-01-15 WO disclosed