SCHEMBL8090953

SCHEMBL8090953

CC(C)(C)OC(=O)CN(CCN(CC(=O)OC(C)(C)C)CC(Cc1ccccc1)N(CC(=O)OC(C)(C)C)CC(=O)OC(C)(C)C)CC(=O)OC(C)(C)C

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATM Q13315 1/20 0.39
ITGA4 P13612 1/20 0.38
ITGB7 P26010 1/20 0.38
AKT1 P31749 2/20 0.38
CTSS P25774 2/20 0.37
CTSL P07711 1/20 0.37
CTSB P07858 1/20 0.37
CTSK P43235 1/20 0.37
ACE P12821 1/20 0.36
MEN1 O00255 1/20 0.36
LMNA P02545 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
ALOX15 P16050 1/20 0.36
TSHR P16473 1/20 0.36
CYP2C19 P33261 1/20 0.36
SCN1A P35498 1/20 0.36
KMT2A Q03164 1/20 0.36
HIF1A Q16665 1/20 0.36
SCN2A Q99250 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5374479 0.89 CTSS (0.38) CTSSCTSKOPRM1OPRD1OPRK1
SCHEMBL3748687 0.88 NR1D1 (0.36) CTSSCTSKNR1D1
SCHEMBL8957471 0.87 CA1 (0.38) CTSSCTSKOPRM1OPRD1OPRK1
SCHEMBL8084139 0.86 PPARA (0.43) CTSSMAOBNPSR1
SCHEMBL9137645 0.86 MAOB (0.44) ATMLMNAOPRM1OPRD1OPRK1
SCHEMBL8099592 0.86 SMN1; SMN2 (0.40) TSHRMAOBNR1D1
SCHEMBL5033940 0.85 NR1D1 (0.36) ATMAKT1CTSSCTSLCTSB
SCHEMBL7516386 0.85 PTPN1 (0.41) MEN1KMT2AMAOBNR1D1
SCHEMBL92706 0.85 ACACB (0.38) ATMLMNANR1D1
SCHEMBL15044629 0.85 ACACB (0.38) ATMLMNANR1D1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6039931-A Derivatized DTPA complexes, pharmaceutical agents containing these compounds, their use, and processes for their production SCHERING AKTIENGESELLSCHAFT (DE) 2000-03-21 US disclosed
US-5798092-A METAL COMPLEXES; CONTRAST AGENTS FOR MEDICAL IMAGING SCHERING AKTIENGESELLSCHAFT (DE) 1998-08-25 US disclosed
US-5695739-A Derivatized DTPA complexes, pharmaceutical agents containing these compounds, their use, and processes for their production SCHERING AKTIENGESELLSCHAFT (DE) 1997-12-09 US disclosed
EP-0405704-B1 DTPA-complexes derivatives, pharmaceutical compositions containing them, their use and process for their preparation SCHERING AG (DE) 1994-12-14 EP disclosed
EP-0405704-A2 DTPA-complexes derivatives, pharmaceutical compositions containing them, their use and process for their preparation SCHERING AKTIENGESELLSCHAFT (DE) 1991-01-02 EP disclosed