SCHEMBL8091032

SCHEMBL8091032

CCC[CH]C(c1ccccc1)N(C)CCCc1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 8/20 0.50
SLC6A2 P23975 2/20 0.49
SLC6A4 P31645 2/20 0.49
SLC6A3 Q01959 2/20 0.49
KCNH2 Q12809 2/20 0.49
CHRM2 P08172 1/20 0.49
HTR1A P08908 1/20 0.49
ADRA2A P08913 1/20 0.49
CHRM1 P11229 1/20 0.49
DRD1 P21728 1/20 0.49
ADRA1A P35348 1/20 0.49
OPRM1 P35372 1/20 0.49
DRD3 P35462 1/20 0.49
AOC3 Q16853 1/20 0.45
BCHE P06276 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8084439 0.78 AOC3 (0.39) SIGMAR1AOC3
SCHEMBL11135639 0.75 SIGMAR1 (0.54) SIGMAR1SLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL14424026 0.71 SIGMAR1 (0.71) SIGMAR1SLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL8091279 0.70 SIGMAR1 (0.50) SIGMAR1KCNH2
SCHEMBL11643972 0.69 SIGMAR1 (0.64) SIGMAR1SLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL12540441 0.69 OPRM1 (0.74) SLC6A2SLC6A4SLC6A3KCNH2CHRM2
SCHEMBL10991198 0.69 KCNH2 (0.43) SIGMAR1KCNH2OPRM1DRD3
SCHEMBL988251 0.69 KCNH2 (0.43) SIGMAR1KCNH2OPRM1DRD3
SCHEMBL8091031 0.69 SIGMAR1 (0.62) SIGMAR1SLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL9373860 0.69 SIGMAR1 (0.52) SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6057371-A TREATMENT OF CENTRAL NERVOUS SYSTEM DISORDERS, GASTROINTESTINAL DISORDERS, DRUG ABUSE, ANGINA, MIGRAINE, HYPERTENSION AND DEPRESSION VIRGINIA COMMONWEALTH UNIVERSITY (US) 2000-05-02 US claimed
EP-0591426-A1 SIGMA RECEPTOR LIGANDS AND THE USE THEREOF VIRGINIA COMMONWEALTH UNIVERSITY (US) 1994-04-13 EP claimed
WO-1993000313-A2 SIGMA RECEPTOR LIGANDS AND THE USE THEREOF VIRGINIA COMMONWEALTH UNIVERSITY (US) 1993-01-07 WO claimed