SCHEMBL8091176

SCHEMBL8091176

O=C(O)c1cn(C2COC2)c2c(Cl)c(F)c(F)cc2c1=O

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.54
POLB P06746 2/20 0.54
CHRM2 P08172 1/20 0.54
CHRM1 P11229 1/20 0.54
OPRM1 P35372 1/20 0.54
OPRD1 P41143 1/20 0.54
TOP2A P11388 8/20 0.52
TOP2B Q02880 8/20 0.52
KDM4E B2RXH2 6/20 0.45
KMT2A Q03164 1/20 0.45
HPGD P15428 2/20 0.45
HSD17B10 Q99714 2/20 0.45
ALB P02768 1/20 0.45
HRH3 Q9Y5N1 1/20 0.45
AADAT Q8N5Z0 2/20 0.44
TUBB4A P04350 1/20 0.44
TUBB P07437 1/20 0.44
TUBA3C P0DPH7 1/20 0.44
TUBA1B P68363 1/20 0.44
TUBA4A P68366 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL500386 0.89 ALDH1A1 (0.66) ALDH1A1POLBCHRM2CHRM1OPRM1
SCHEMBL29962586 0.89 ALDH1A1 (0.66) ALDH1A1POLBCHRM2CHRM1OPRM1
SCHEMBL8136160 0.89 TOP2A (0.57) ALDH1A1POLBCHRM2CHRM1OPRM1
SCHEMBL9272261 0.88 TOP2A (0.54) ALDH1A1POLBCHRM2CHRM1OPRM1
Fluoride SCHEMBL5143354 0.87 ALDH1A1 (0.63) ALDH1A1POLBCHRM2CHRM1OPRM1
SCHEMBL5143359 0.86 ALDH1A1 (0.62) ALDH1A1POLBCHRM2CHRM1OPRM1
SCHEMBL9045760 0.85 ALDH1A1 (0.41) ALDH1A1POLBCHRM2CHRM1OPRM1
SCHEMBL9265070 0.84 ADRB2 (0.52) ALDH1A1POLBCHRM2CHRM1OPRM1
SCHEMBL9266603 0.83 KDM4E (0.55) ALDH1A1POLBOPRM1TOP2ATOP2B
SCHEMBL9267055 0.82 KDM4E (0.64) ALDH1A1POLBCHRM2CHRM1OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6018054-A INTERMEDIATE COMPOUNDS FOR PREPARING NOVEL QUINOLONE AND NAPHTHYRIDONE DERIVATIVES WHICH ARE SUBSTITUTED IN THE 7-POSITION BY A PARTIALLY HYDROGENATED ISOINDOLINYL RING, USE AS ANTIBACTERIAL AGENTS AND AS FEED ADDITIVES BAYER AKTIENGESELLSCHAFT (DE) 2000-01-25 US disclosed
US-5739339-A BACTERICIDES, ANTIPROTOZOA AGENTS BAYER AKTIENGESELLSCHAFT (DE) 1998-04-14 US disclosed
US-5556979-A ANIMAL FEEDS BAYER AKTIENGESELLSCHAFT (DE) 1996-09-17 US disclosed
EP-0588166-B1 Antibacterial 7-isoindolinyl-quinolone and naphthyridone derivatives BAYER AG (DE) 1996-06-05 EP disclosed
US-5407932-A Bactericides WAKUNAGA SEIYAKU KABUSHIKI KAISHA (JP) 1995-04-18 US disclosed
EP-0393400-B1 Novel quinolone derivatives, preparation processes thereof, and antibacterial agents containing the same WAKUNAGA SEIYAKU KK (JP) 1994-12-21 EP disclosed
EP-0588166-A2 Antibacterial 7-isoindolinyl-quinolone and naphthyridone derivatives BAYER AG (DE) 1994-03-23 EP disclosed
US-5245037-A Synthetic bactericides WAKUNAGA SEIYAKU KABUSHIKI KAISHA (JP) 1993-09-14 US disclosed
EP-0393400-A1 Novel quinolone derivatives, preparation processes thereof, and antibacterial agents containing the same WAKUNAGA SEIYAKU KABUSHIKI KAISHA (JP) 1990-10-24 EP disclosed