SCHEMBL8092353

SCHEMBL8092353

Cc1ccc2c(c1[N+](=O)[O-])C(=O)NC2=O

nearest known ligand 0.55

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.55
TSHR P16473 4/20 0.55
CYP3A4 P08684 2/20 0.55
TDP1 Q9NUW8 3/20 0.46
PARP1 P09874 2/20 0.40
POLB P06746 1/20 0.40
SMN1; SMN2 Q16637 2/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
MAOA P21397 1/20 0.38
MAOB P27338 1/20 0.38
MAPT P10636 1/20 0.37
CASP3 P42574 2/20 0.36
TDP2 O95551 1/20 0.36
PPOX P50336 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9503458 0.81 CYP3A4 (0.51) TSHRCYP3A4TDP1PARP1POLB
SCHEMBL28138230 0.79 CYP3A4 (0.46) ALDH1A1TSHRCYP3A4TDP1PARP1
SCHEMBL10785547 0.78 TSHR (0.83) ALDH1A1TSHRCYP3A4TDP1SMN1; SMN2
SCHEMBL5151002 0.77 POLB (0.44) ALDH1A1TSHRCYP3A4TDP1PARP1
SCHEMBL8098610 0.76 TDP1 (0.46) TSHRCYP3A4TDP1PARP1POLB
SCHEMBL13058018 0.75 ALDH1A1 (0.50) ALDH1A1TSHRCYP3A4TDP1SMN1; SMN2
SCHEMBL8098589 0.74 TDP1 (0.39) ALDH1A1TSHRCYP3A4TDP1PARP1
SCHEMBL32680469 0.74 TDP2 (0.56) ALDH1A1PARP1POLBMAOAMAOB
SCHEMBL10962827 0.74 TDP2 (0.56) ALDH1A1PARP1POLBMAOAMAOB
SCHEMBL19585641 0.72 ALDH1A1 (0.59) ALDH1A1TSHRCYP3A4TDP1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106459412-B Fibre-reinforced polyetherimide compositions 沙特基础工业全球技术公司 2019-07-30 CN disclosed
CN-107246369-B Compressor including polymerizing component 沙特基础全球技术有限公司 2019-07-12 CN disclosed
CN-104641424-B Polymer nanocomposite for electronic application 沙特基础全球技术有限公司 2017-08-25 CN disclosed
EP-2994919-A2 DUAL LAYER WIRE COATINGS SABIC Global Technologies B.V. (NL) 2016-03-16 EP disclosed
WO-2014183011-A2 DUAL LAYER WIRE COATINGS SABIC INNOVATIVE PLASTICS IP B.V. (NL) 2014-11-13 WO disclosed
EP-2773686-A1 STEAM PURIFICATION OF POLYIMIDE RESINS SABIC Innovative Plastics IP B.V. (NL) 2014-09-10 EP disclosed
EP-2773685-A1 SOLVENTLESS PROCESS FOR THE PREPARATION OF AMINE FUNCTIONAL POLYETHERIMIDE RESINS WITH IMPROVED MELT FLOW SABIC Innovative Plastics IP B.V. (NL) 2014-09-10 EP disclosed
WO-2013066791-A1 STEAM PURIFICATION OF POLYIMIDE RESINS SABIC INNOVATIVE PLASTICS IP B.V. (NL) 2013-05-10 WO disclosed
WO-2013066783-A1 SOLVENTLESS PROCESS FOR THE PREPARATION OF AMINE FUNCTIONAL POLYETHERIMIDE RESINS WITH IMPROVED MELT FLOW SABIC INNOVATIVE PLASTICS IP B.V. (NL) 2013-05-10 WO disclosed
EP-1059291-A2 Process for preparing bis(ether anhydrides) GENERAL ELECTRIC COMPANY (US) 2000-12-13 EP disclosed
US-6008374-A REACTING N-ALKYL NITROPHTHALIMIDE AND A BISPHENOL ALKALI METAL SALT TO FORM BISIMIDE, EXTRACTING THE FORMED BISIMIDE GENERAL ELECTRIC COMPANY (US) 1999-12-28 US disclosed
US-5936099-A N-ALKYL PHTHALAMIDES BY REACTING LIQUID (C3-C6)ALKYLAMINES AND PHTHALIC ANHYDRIDE; NITRATION FOLLOWED BY REACTING WITH A BISPHENOL A; EXCHANGE REACTION TO FORM DIANHYDRIDE; HYDROLYSIS TO PRODUCE TETRACID MONOMER FOR POLYETHERIMIDES GENERAL ELECTRIC CO. (US) 1999-08-10 US disclosed
US-5719295-A FROM N-ALKYL NITROPHTHALAMIDE GENERAL ELECTRIC COMPANY (US) 1998-02-17 US disclosed
US-5536846-A NITRATION, PURIFICATION, LIQUID EXTRACTION, DRYING AND PURIFICATION THEN REACTION WITH ALKALI METAL BISPHENOL AND TRANSFORMATION GENERAL ELECTRIC COMPANY (US) 1996-07-16 US disclosed
EP-0684232-A1 Process for preparing bis(ether anhydrides) GENERAL ELECTRIC COMPANY (US) 1995-11-29 EP disclosed