SCHEMBL8092829

SCHEMBL8092829

COc1cccc(CNc2nc(-c3ccc(F)cc3)c(-c3ccc(S(C)(=O)=O)cc3)cc2C#N)c1

nearest known ligand 0.51

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 11/20 0.51
MAPT P10636 1/20 0.49
PTGS1 P23219 2/20 0.43
MAPK8 P45983 1/20 0.43
MAPK9 P45984 1/20 0.43
MAPK10 P53779 1/20 0.43
HIF1A Q16665 1/20 0.43
CNR1 P21554 1/20 0.42
SQOR Q9Y6N5 1/20 0.41
TNF P01375 1/20 0.41
PDE4B Q07343 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8099660 0.92 MAPT (0.49) PTGS2MAPTPTGS1HIF1ACNR1
SCHEMBL8099266 0.84 PTGS2 (0.53) PTGS2PTGS1MAPK8MAPK9
SCHEMBL8101771 0.83 PTGS2 (0.54) PTGS2PTGS1CNR1
SCHEMBL8101829 0.82 PTGS2 (0.52) PTGS2PTGS1
SCHEMBL8093657 0.82 PTGS2 (0.56) PTGS2PTGS1MAPK8MAPK9MAPK10
SCHEMBL8099373 0.82 PTGS2 (0.51) PTGS2PTGS1MAPK8MAPK9MAPK10
SCHEMBL8419819 0.81 MAPT (0.48) MAPTHIF1A
SCHEMBL8095004 0.81 PTGS2 (0.49) PTGS2PTGS1
SCHEMBL8094067 0.79 PTGS2 (0.49) PTGS2PTGS1CNR1
SCHEMBL8095119 0.79 HPGD (0.47) PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0808304-B1 2,3-SUBSTITUTED PYRIDINES FOR THE TREATMENT OF INFLAMMATION SEARLE & CO (US) 2000-12-27 EP disclosed
US-5916905-A ANTIARTHRITIC AGENTS; ANALGESICS; ANTIPYRETICS G. D. SEARLE & CO. (US) 1999-06-29 US disclosed
US-5686470-A 2, 3-substituted pyridines for the treatment of inflammation WEIER RICHARD M (US) 1997-11-11 US disclosed