SCHEMBL8095004

SCHEMBL8095004

CS(=O)(=O)c1ccc(-c2cc(C#N)c(NCc3ccco3)nc2-c2ccc(F)cc2)cc1

nearest known ligand 0.49

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 15/20 0.49
KDM4E B2RXH2 3/20 0.48
ALDH1A1 P00352 1/20 0.48
GAA P10253 1/20 0.48
CASP1 P29466 1/20 0.48
HSD17B10 Q99714 1/20 0.48
EED O75530 2/20 0.44
ADRA2A P08913 1/20 0.44
ADRA2C P18825 1/20 0.44
PDE4D Q08499 1/20 0.44
RBBP4 Q09028 1/20 0.44
SUZ12 Q15022 1/20 0.44
EZH2 Q15910 1/20 0.44
PTGS1 P23219 3/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8086615 0.91 PTGS2 (0.49) PTGS2KDM4EALDH1A1GAACASP1
SCHEMBL8095250 0.84 PTGS2 (0.49) PTGS2PTGS1
SCHEMBL8101829 0.84 PTGS2 (0.52) PTGS2PTGS1
SCHEMBL8099266 0.83 PTGS2 (0.53) PTGS2ALDH1A1PTGS1
SCHEMBL8101771 0.83 PTGS2 (0.54) PTGS2PTGS1
SCHEMBL8099373 0.82 PTGS2 (0.51) PTGS2PTGS1
SCHEMBL8092829 0.81 PTGS2 (0.51) PTGS2PTGS1
SCHEMBL8094067 0.81 PTGS2 (0.49) PTGS2PTGS1
SCHEMBL8095119 0.81 HPGD (0.47) PTGS2KDM4EALDH1A1PTGS1
SCHEMBL8093657 0.80 PTGS2 (0.56) PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0808304-B1 2,3-SUBSTITUTED PYRIDINES FOR THE TREATMENT OF INFLAMMATION SEARLE & CO (US) 2000-12-27 EP disclosed
US-5916905-A ANTIARTHRITIC AGENTS; ANALGESICS; ANTIPYRETICS G. D. SEARLE & CO. (US) 1999-06-29 US disclosed
US-5686470-A 2, 3-substituted pyridines for the treatment of inflammation WEIER RICHARD M (US) 1997-11-11 US disclosed