SCHEMBL8092840

SCHEMBL8092840

CCOC(=O)NC1CC=CC2CN(c3cc4c(cc3F)c(=O)c(C(=O)O)cn4C(C)(C)C)CC21

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 7/20 0.41
ALDH1A1 P00352 9/20 0.40
DRD3 P35462 1/20 0.40
KDM4E B2RXH2 10/20 0.40
HPGD P15428 7/20 0.40
LMNA P02545 4/20 0.40
MAPT P10636 2/20 0.40
HTT P42858 3/20 0.40
TSHR P16473 2/20 0.40
BRD4 O60885 1/20 0.40
CYP2J2 P51589 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
NPC1 O15118 1/20 0.39
USP2 O75604 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
TP53 P04637 1/20 0.37
POLB P06746 1/20 0.37
GAA P10253 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9045440 0.91 ALDH1A1 (0.35) HSD17B10ALDH1A1DRD3KDM4EHPGD
SCHEMBL8083248 0.89 DRD3 (0.53) HSD17B10ALDH1A1DRD3KDM4EHPGD
SCHEMBL8092868 0.88 KDM4E (0.55) HSD17B10ALDH1A1KDM4EHPGDLMNA
SCHEMBL8091199 0.82 ALDH1A1 (0.44) HSD17B10ALDH1A1DRD3KDM4EHPGD
SCHEMBL9046354 0.82 KDM4E (0.44) HSD17B10ALDH1A1DRD3KDM4EHPGD
SCHEMBL9045493 0.81 KDM4E (0.44) HSD17B10ALDH1A1KDM4EHPGDLMNA
SCHEMBL8084270 0.79 HSD17B10 (0.53) HSD17B10ALDH1A1DRD3KDM4EHPGD
SCHEMBL9095828 0.78 KCNH2 (0.48) HSD17B10ALDH1A1KDM4EHPGDLMNA
SCHEMBL8083134 0.78 KCNH2 (0.42) HSD17B10ALDH1A1KDM4EHPGDMEN1
SCHEMBL8091409 0.77 KDM4E (0.40) HSD17B10ALDH1A1KDM4EHPGDLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6018054-A INTERMEDIATE COMPOUNDS FOR PREPARING NOVEL QUINOLONE AND NAPHTHYRIDONE DERIVATIVES WHICH ARE SUBSTITUTED IN THE 7-POSITION BY A PARTIALLY HYDROGENATED ISOINDOLINYL RING, USE AS ANTIBACTERIAL AGENTS AND AS FEED ADDITIVES BAYER AKTIENGESELLSCHAFT (DE) 2000-01-25 US disclosed
US-5556979-A ANIMAL FEEDS BAYER AKTIENGESELLSCHAFT (DE) 1996-09-17 US disclosed