SCHEMBL8093673

SCHEMBL8093673

CCc1cc(Cl)ccc1N=C=O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 2/20 0.48
GABRB2 P47870 2/20 0.48
CYP3A4 P08684 4/20 0.40
TDP1 Q9NUW8 2/20 0.40
HPGD P15428 2/20 0.40
ALDH1A1 P00352 1/20 0.40
TRPA1 O75762 1/20 0.38
MAPK1 P28482 2/20 0.36
SLC6A4 P31645 5/20 0.35
SLC6A2 P23975 4/20 0.35
FLT1 P17948 1/20 0.35
FLT4 P35916 1/20 0.35
KDR P35968 1/20 0.35
LMNA P02545 2/20 0.34
MEN1 O00255 1/20 0.34
SLC22A1 O15245 1/20 0.34
USP2 O75604 1/20 0.34
HSP90AA1 P07900 1/20 0.34
MAPT P10636 1/20 0.34
HSPD1 P10809 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10885131 0.87 MAPK1 (0.37) GABRA1GABRB2CYP3A4TDP1HPGD
SCHEMBL27609924 0.84 CYP2A6 (0.38) GABRA1GABRB2CYP3A4TDP1HPGD
SCHEMBL14008752 0.84 GABRA1 (0.50) GABRA1GABRB2CYP3A4TDP1HPGD
SCHEMBL11464398 0.84 TDP1 (0.35) GABRA1GABRB2CYP3A4TDP1HPGD
SCHEMBL894932 0.81 CYP3A4 (0.55) GABRA1GABRB2CYP3A4TDP1HPGD
SCHEMBL7704447 0.80 CYP3A4 (0.33) GABRA1GABRB2CYP3A4TDP1HPGD
SCHEMBL109348 0.79 CYP3A4 (0.56) GABRA1GABRB2CYP3A4TDP1HPGD
SCHEMBL11509013 0.79 GABRA1 (0.46) GABRA1GABRB2CYP3A4TDP1HPGD
SCHEMBL28222905 0.79 GABRA1 (0.46) GABRA1GABRB2CYP3A4TDP1HPGD
SCHEMBL11862224 0.78 GABRA1 (0.46) GABRA1GABRB2CYP3A4HPGDTRPA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0973936-A1 COMBINATORIAL LIBRARIES OF PEPTIDOMIMETIC AMINOTHIOETHER ACIDS ELI LILLY AND COMPANY (US) 2000-01-26 EP disclosed
WO-1998046786-A1 COMBINATORIAL LIBRARIES OF PEPTIDOMIMETIC AMINOTHIOETHER ACIDS ELI LILLY AND COMPANY (US) 1998-10-22 WO disclosed
US-4174398-A Combating fungi with 1-alkyl-1-(1,3,4-thiadiazol-2-yl)-3-phenyl-ureas BAYER AKTIENGESELLSCHAFT (DE) 1979-11-13 US disclosed
US-4163112-A INSECTICIDES VELSICOL CHEMICAL CORPORATION (US) 1979-07-31 US disclosed