SCHEMBL8094722

SCHEMBL8094722

C=C(C)c1nc(N)ccc1OC

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 1/20 0.43
NCF1 P14598 1/20 0.36
KDM4E B2RXH2 4/20 0.34
L3MBTL1 Q9Y468 3/20 0.34
MAPT P10636 3/20 0.34
THRB P10828 2/20 0.34
NPC1 O15118 2/20 0.34
MAPK1 P28482 2/20 0.34
RAB9A P51151 2/20 0.34
GAA P10253 1/20 0.34
BLM P54132 1/20 0.34
ATM Q13315 1/20 0.34
ALDH1A1 P00352 4/20 0.33
LMNA P02545 3/20 0.33
PDE10A Q9Y233 1/20 0.33
NQO2 P16083 1/20 0.33
PDE4A P27815 1/20 0.33
PDE4B Q07343 1/20 0.33
PDE4C Q08493 1/20 0.33
PDE4D Q08499 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15099897 0.79 KDM4E (0.37) KDM4EL3MBTL1MAPTNPC1MAPK1
SCHEMBL2273523 0.74 NQO1 (0.41) KDM4EALDH1A1PDE10APDE4APDE4B
SCHEMBL18560621 0.74 KDM4E (0.33) KDM4EL3MBTL1MAPTALDH1A1NQO2
SCHEMBL15090987 0.73 NOS3 (0.34) KDM4ENPC1RAB9AGAAALDH1A1
SCHEMBL15091095 0.71 MEN1 (0.42) KDM4EL3MBTL1MAPTNPC1RAB9A
SCHEMBL9810196 0.71 MCHR1 (0.52) MCHR1NCF1KDM4EL3MBTL1MAPT
SCHEMBL15091050 0.70 POLB (0.40) MCHR1NCF1KDM4EMAPTNPC1
SCHEMBL22222454 0.70 KDM4E (0.40) MCHR1KDM4EL3MBTL1MAPTTHRB
SCHEMBL26137569 0.70 GABRP (0.42) ALDH1A1LMNANOS1NOS3NOS2
SCHEMBL359862 0.70 MCHR1 (0.50) MCHR1NCF1KDM4EL3MBTL1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009020642-A1 PYRIDINE CARBOXAMIDE OREXIN RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 2009-02-12 WO disclosed