SCHEMBL8094825

SCHEMBL8094825

COC(=O)CSC1CC(=O)N1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.37
SMN1; SMN2 Q16637 3/20 0.37
MAPK1 P28482 1/20 0.37
POLB P06746 1/20 0.36
ITGB1 P05556 2/20 0.36
ITGA5 P08648 2/20 0.36
ITGB3 P05106 1/20 0.36
ITGB2 P05107 1/20 0.36
ITGAV P06756 1/20 0.36
ITGA2B P08514 1/20 0.36
ITGB5 P18084 1/20 0.36
ITGAL P20701 1/20 0.36
BRD4 O60885 1/20 0.36
GAA P10253 1/20 0.35
TDP1 Q9NUW8 3/20 0.35
TP53 P04637 2/20 0.34
PKM P14618 1/20 0.34
TSHR P16473 1/20 0.34
LMNA P02545 2/20 0.34
MAPT P10636 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11262107 0.77 ITGB1 (0.36) ALDH1A1SMN1; SMN2MAPK1ITGB1ITGA5
SCHEMBL11262117 0.77 ITGB1 (0.36) ALDH1A1SMN1; SMN2MAPK1ITGB1ITGA5
SCHEMBL8102643 0.76 TSHR (0.37) ALDH1A1SMN1; SMN2ITGB1ITGA5ITGB3
SCHEMBL10948404 0.75 TSHR (0.42) ALDH1A1ITGB1ITGA5ITGB3ITGB2
SCHEMBL10948414 0.75 TSHR (0.42) ALDH1A1ITGB1ITGA5ITGB3ITGB2
SCHEMBL9836292 0.72 ITGB1 (0.59) ITGB1ITGA5ITGB3ITGB2ITGAV
SCHEMBL10968083 0.72 ITGB1 (0.59) ITGB1ITGA5ITGB3ITGB2ITGAV
SCHEMBL9836299 0.72 ITGB1 (0.59) ITGB1ITGA5ITGB3ITGB2ITGAV
SCHEMBL10814097 0.69 TSHR (0.46) ALDH1A1MAPK1ITGB1ITGA5ITGB3
SCHEMBL11169353 0.68 ITGB1 (0.36) ITGB1ITGA5ITGB3ITGB2ITGAV

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6071899-A Azetidinone derivatives for the treatment of atherosclerosis SMITHKLINE BEECHAM P.L.C. (GB) 2000-06-06 US disclosed
EP-0788478-A1 AZETIDINONE DERIVATIVES FOR THE TREATMENT OF ATHEROSCLEROSIS SMITHKLINE BEECHAM PLC (GB) 1997-08-13 EP disclosed
WO-1996013484-A1 AZETIDINONE DERIVATIVES FOR THE TREATMENT OF ATHEROSCLEROSIS SMITHKLINE BEECHAM PLC (GB) 1996-05-09 WO disclosed
EP-0053815-B1 2-OXOAZETIDINE DERIVATIVES, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 1985-05-08 EP disclosed