SCHEMBL8094981

SCHEMBL8094981

COc1ccc(CS[C@H]2C[C@@H](C(=O)N3CC[C@H](NC(=O)C4CCCCN4C(=O)OCc4ccc([N+](=O)[O-])cc4)C3)N(C(=O)OCc3ccc([N+](=O)[O-])cc3)C2)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.40
NPSR1 Q6W5P4 1/20 0.40
TP53 P04637 1/20 0.40
CTSB P07858 1/20 0.38
CTSS P25774 1/20 0.38
CTSK P43235 1/20 0.38
LMNA P02545 2/20 0.37
KDM4E B2RXH2 1/20 0.37
GAA P10253 1/20 0.36
MAPT P10636 2/20 0.36
HPGD P15428 1/20 0.36
MMP1 P03956 1/20 0.36
MMP2 P08253 1/20 0.36
MMP3 P08254 1/20 0.36
MMP7 P09237 1/20 0.36
MMP9 P14780 1/20 0.36
MMP8 P22894 1/20 0.36
MAPK1 P28482 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
MEN1 O00255 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7458116 0.98 ALDH1A1 (0.42) ALDH1A1NPSR1TP53CTSKLMNA
SCHEMBL7458108 0.98 ALDH1A1 (0.42) ALDH1A1NPSR1TP53CTSKLMNA
SCHEMBL8095066 0.94 ALDH1A1 (0.43) ALDH1A1NPSR1TP53CTSKLMNA
SCHEMBL8095064 0.94 ALDH1A1 (0.43) ALDH1A1NPSR1TP53CTSKLMNA
SCHEMBL8435157 0.91 SMN1; SMN2 (0.45) ALDH1A1GAAMAPTMMP1MMP2
SCHEMBL8436042 0.91 SMN1; SMN2 (0.45) ALDH1A1GAAMAPTMMP1MMP2
SCHEMBL8438094 0.91 ALDH1A1 (0.44) ALDH1A1NPSR1TP53GAAMAPT
SCHEMBL8438096 0.91 ALDH1A1 (0.44) ALDH1A1NPSR1TP53GAAMAPT
SCHEMBL8436455 0.88 GAA (0.40) ALDH1A1GAAMAPTMMP1MMP2
SCHEMBL8435165 0.88 ALDH1A1 (0.43) ALDH1A1LMNAGAAMAPTMMP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008115381-A1 PYRIDAZINONE DERIVATIVES USEFUL AS GLUCAN SYNTHASE INHIBITORS SCHERING CORPORATION (US) 2008-09-25 WO disclosed
US-6090802-A BACTERICIDE SANKYO COMPANY, LIMITED (JP) 2000-07-18 US disclosed
EP-0882728-A1 1-METHYLCARBAPENEM DERIVATIVES SANKYO COMPANY LIMITED (JP) 1998-12-09 EP disclosed